SCHEMBL8430503

SCHEMBL8430503

CCCc1cc(Cl)c(C(=O)NC(=N)N)cc1C(F)(F)F

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
RAB9A P51151 1/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2D6 P10635 2/20 0.33
CYP2C19 P33261 2/20 0.33
JUN P05412 1/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
MEN1 O00255 1/20 0.33
CYP2C9 P11712 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33
POLB P06746 2/20 0.33
APEX1 P27695 1/20 0.33
TDP1 Q9NUW8 2/20 0.32
AR P10275 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8335175 0.99 SMN1; SMN2 (0.33) SMN1; SMN2TP53MAPTRAB9ACYP1A2
SCHEMBL8428726 0.81 TP53 (0.39) SMN1; SMN2TP53MAPTRAB9APOLB
Hydrochloric Acid SCHEMBL8337102 0.80 TP53 (0.38) SMN1; SMN2TP53MAPTRAB9APOLB
SCHEMBL8426433 0.80 POLB (0.38) SMN1; SMN2TP53MAPTRAB9APOLB
SCHEMBL7797854 0.79 TMPRSS4 (0.41) SMN1; SMN2TP53MAPTRAB9ACYP1A2
Hydrochloric Acid SCHEMBL8332842 0.79 POLB (0.38) SMN1; SMN2TP53MAPTRAB9APOLB
SCHEMBL8332877 0.78 CFTR (0.42) MAPTCYP1A2CYP2C19HTTEPHX2
Hydrochloric Acid SCHEMBL7791912 0.78 TMPRSS4 (0.40) SMN1; SMN2TP53MAPTRAB9ACYP1A2
SCHEMBL8426429 0.78 JUN (0.39) JUNNFKB1NFKB2RELAPOLB
SCHEMBL8428710 0.78 MAPT (0.40) MAPTRAB9AMEN1HTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0791577-B1 Ortho-substituted benzylguanidines, process for their preparation and their use as medicament or diagnostic agent as well as medicament containing them HOECHST AG (DE) 1999-11-03 EP claimed