SCHEMBL8429637

SCHEMBL8429637

O=C(CC(c1ccccc1)c1ccccc1)N1CCN(C(c2ccc(O)cc2)c2ccc3c(c2)OCO3)CC1

nearest known ligand 0.92

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 15/20 0.65
CACNB1 Q02641 15/20 0.65
CACNA1B Q00975 13/20 0.65
CACNA1C Q13936 11/20 0.65
CACNA1H O95180 1/20 0.65
CACNA1G O43497 3/20 0.60
CACNA1A O00555 3/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5267438 0.96 CACNA2D1 (0.70) CACNA2D1CACNB1CACNA1BCACNA1CCACNA1H
SCHEMBL8446337 0.88 CACNA2D1 (0.77) CACNA2D1CACNB1CACNA1BCACNA1CCACNA1H
SCHEMBL5266285 0.87 CACNA2D1 (0.86) CACNA2D1CACNB1CACNA1BCACNA1CCACNA1H
SCHEMBL5549190 0.81 CACNA2D1 (0.73) CACNA2D1CACNB1CACNA1BCACNA1CCACNA1H
Z160 SCHEMBL4180792 0.80 CACNA2D1 (1.00) CACNA2D1CACNB1CACNA1BCACNA1CCACNA1H
SCHEMBL15266877 0.78 SMAD3 (0.60)
SCHEMBL3395399 0.78 CACNA2D1 (0.71) CACNA2D1CACNB1CACNA1BCACNA1C
SCHEMBL5270085 0.77 CACNA2D1 (0.77) CACNA2D1CACNB1CACNA1BCACNA1CCACNA1H
SCHEMBL5266301 0.76 CACNA2D1 (1.00) CACNA2D1CACNB1CACNA1BCACNA1CCACNA1H
SCHEMBL5268519 0.76 CACNA2D1 (1.00) CACNA2D1CACNB1CACNA1BCACNA1CCACNA1H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040259866-A1 Calcium channel blockers comprising two benzhydril moieties ZALICUS PHARMACEUTICALS LTD. (CA) 2004-12-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040259866-A1 Calcium channel blockers comprising two benzhydril moieties CACNA1C, CACNA1F, CACNA1D CACNA2D1 41/4885CACNB1 14/4885CACNA1B 4/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.