SCHEMBL8430347

SCHEMBL8430347

N[C@@H](c1ccc(C(F)(F)F)cc1)[C@@H](O)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.50
CES1 P23141 2/20 0.50
GRM8 O00222 1/20 0.50
GRM4 Q14833 1/20 0.50
KIF11 P52732 1/20 0.44
ACP3 P15309 1/20 0.44
GRIK1 P39086 1/20 0.43
GRIK2 Q13002 1/20 0.43
SLC1A3 P43003 1/20 0.43
SLC1A2 P43004 1/20 0.43
SLC1A1 P43005 1/20 0.43
AKR1C3 P42330 2/20 0.42
AKR1C2 P52895 2/20 0.42
HSD11B1 P28845 1/20 0.42
SRD5A2 P31213 1/20 0.42
CNR2 P34972 2/20 0.41
PDPK1 O15530 1/20 0.41
GSK3B P49841 1/20 0.41
FFAR1 O14842 1/20 0.39
PSEN1 P49768 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5597212 0.84 PDPK1 (0.49) CES2CES1GRM8GRM4KIF11
Cadaverine Tartrate SCHEMBL10560377 0.83 PDE2A (0.50) CES2CES1GRM8GRM4KIF11
SCHEMBL11902072 0.79 GRM8 (0.50) CES2CES1GRM8GRM4KIF11
SCHEMBL5225725 0.79 GRM8 (0.50) CES2CES1GRM8GRM4KIF11
SCHEMBL8426162 0.79 HDAC3 (0.41) GRIK1GRIK2SLC1A3SLC1A2SLC1A1
SCHEMBL18125936 0.79 GRM8 (0.50) CES2CES1GRM8GRM4KIF11
SCHEMBL5018968 0.79 NR1I2 (0.53) CES2CES1GRM8GRM4KIF11
SCHEMBL4967991 0.79 NR1I2 (0.53) CES2CES1GRM8GRM4KIF11
SCHEMBL15137434 0.78 KIF11 (0.46) CES2CES1KIF11ACP3
SCHEMBL15670412 0.78 KIF11 (0.46) CES2CES1KIF11ACP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5939561-A Process for the preparation of β-phenylisoserine and β-lactam and their analogues RHONE-POULENCE RORER S.A. (FR) 1999-08-17 US disclosed
US-5763628-A Process for the preparation of β-phenylisoserine and its analogues RHONE-POULENCE RORER S.A. (FR) 1998-06-09 US disclosed
US-5608102-A Process for the preparation of β-phenylisoserine and its analogues RHONE-POULENC RORER S.A. (FR) 1997-03-04 US disclosed