SCHEMBL8432173

SCHEMBL8432173

CCc1cc(C(O)(C(=O)O)C(=O)O)ccc1N

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.40
ESR2 Q92731 4/20 0.40
ALDH1A1 P00352 5/20 0.39
MAPT P10636 3/20 0.39
POLB P06746 1/20 0.39
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
CYP1A2 P05177 1/20 0.37
AR P10275 1/20 0.36
CHEK1 O14757 1/20 0.36
FYN P06241 1/20 0.36
PDGFRB P09619 1/20 0.36
PIM1 P11309 1/20 0.36
FGFR1 P11362 1/20 0.36
FLT1 P17948 1/20 0.36
GRK5 P34947 1/20 0.36
MAP2K2 P36507 1/20 0.36
MAPK8 P45983 1/20 0.36
CDK8 P49336 1/20 0.36
RPS6KA3 P51812 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8436002 0.89 ESR1 (0.35) ESR1ESR2ALDH1A1MAPTKMT2A
SCHEMBL9910783 0.80 ESR1 (0.43) ESR1ESR2ALDH1A1MAPTPOLB
SCHEMBL8432092 0.80 ESR1 (0.46) ESR1ESR2ALDH1A1MAPTPOLB
SCHEMBL9204049 0.80 HTT (0.40) ESR1ESR2ALDH1A1MAPTPOLB
SCHEMBL8431885 0.78 HSD17B10 (0.51) ALDH1A1MAPTPOLBKMT2AMEN1
SCHEMBL7096170 0.76 NR1H2 (0.47) KMT2AMEN1HSD17B10SMN1; SMN2
SCHEMBL9199887 0.76 HTT (0.41) ESR1ESR2ALDH1A1MAPTPOLB
SCHEMBL2997187 0.76 KLF10 (0.46) ESR1ESR2ALDH1A1MAPTPOLB
SCHEMBL11511323 0.76 ALDH1A1 (0.48) ESR1ESR2ALDH1A1MAPTPOLB
SCHEMBL30806220 0.76 KLF10 (0.46) ESR1ESR2ALDH1A1MAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0605404-B1 Polycyclic dyes BASF AG (DE) 1999-12-08 EP disclosed
EP-0363034-B1 Polycyclic dyes ZENECA LTD (GB) 1995-01-04 EP disclosed
EP-0605404-A2 Polycyclic dyes ZENECA LIMITED (GB) 1994-07-06 EP disclosed
EP-0570111-A1 Polycyclic dyes ZENECA LIMITED (GB) 1993-11-18 EP disclosed
US-5212313-A For polyester IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-05-18 US disclosed
US-5183888-A Reacting a phenyl tartronic acid with a dihydrobenzofuran, oxidizing, to get dihydrobenzodifuran IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-02-02 US disclosed
US-5084580-A Aniline dyes for polyester fabrics to give green and blue color IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-01-28 US disclosed
EP-0363034-A2 Polycyclic dyes ZENECA LIMITED (GB) 1990-04-11 EP disclosed