SCHEMBL8432206

SCHEMBL8432206

O=C(CSCCS)NCCNC(=O)Cn1ccnc1[N+](=O)[O-]

nearest known ligand 0.65

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.65
THRB P10828 1/20 0.65
CYP2C19 P33261 1/20 0.65
CYP3A4 P08684 1/20 0.55
CYP2D6 P10635 1/20 0.55
OPRK1 P41145 1/20 0.55
CA12 O43570 5/20 0.53
CA1 P00915 5/20 0.53
CA2 P00918 5/20 0.53
CA9 Q16790 5/20 0.53
KMT2A Q03164 1/20 0.41
ALDH1A1 P00352 2/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 2/20 0.35
TYMP P19971 3/20 0.34
HTT P42858 2/20 0.34
TAAR1 Q96RJ0 1/20 0.34
POLB P06746 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8432208 0.84 LMNA (0.50) LMNATHRBCYP2C19CYP3A4CYP2D6
Etanidazole SCHEMBL4414 0.80 LMNA (1.00) LMNATHRBCYP2C19CYP3A4CYP2D6
Etanidazole SCHEMBL8171462 0.80 LMNA (1.00) LMNATHRBCYP2C19CYP3A4CYP2D6
SCHEMBL8483856 0.79 LMNA (0.58) LMNATHRBCYP2C19CYP3A4CYP2D6
SCHEMBL14499615 0.78 LMNA (0.78) LMNATHRBCYP2C19CYP3A4CYP2D6
Etanidazole SCHEMBL9473771 0.78 LMNA (0.97) LMNATHRBCYP2C19CYP3A4CYP2D6
SCHEMBL368130 0.78 LMNA (0.78) LMNATHRBCYP2C19CYP3A4CYP2D6
SCHEMBL8432165 0.78 LMNA (0.78) LMNATHRBCYP2C19CYP3A4CYP2D6
SCHEMBL15024639 0.77 LMNA (0.80) LMNATHRBCYP2C19CYP3A4CYP2D6
SCHEMBL13065838 0.76 LMNA (0.74) LMNATHRBCYP2C19CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6004531-A LIGANDS FOR RADIOPHARMACEUTICALS; CAPABLE OF CHELATING RADIOMETAL SPECIES AND OF BEING BOUND TO BIOLOGICAL TARGETING MOLECULES NYCOMED AMERSHAM PLC (GB) 1999-12-21 US disclosed
US-5932707-A Thioether-containing metal chelating compounds NYCOMED AMERSHAM PLC (GB) 1999-08-03 US disclosed
WO-1994022816-A1 METAL CHELATING COMPOUNDS AMERSHAM INTERNATIONAL PLC (GB) 1994-10-13 WO disclosed
EP-0618191-A1 Metal chelating compounds AMERSHAM INTERNATIONAL plc (GB) 1994-10-05 EP disclosed