SCHEMBL8433599

SCHEMBL8433599

CC(C)[C@H](N)C(O)c1noc(Cc2c(F)cccc2F)n1

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.33
ABCB1 P08183 1/20 0.32
ABCG2 Q9UNQ0 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 2/20 0.31
LMNA P02545 1/20 0.31
NPC1 O15118 1/20 0.31
GLA P06280 1/20 0.31
RAB9A P51151 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
POLB P06746 1/20 0.30
MAPT P10636 1/20 0.30
KMT2A Q03164 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8435334 0.99 IDH1 (0.33) IDH1ABCB1ABCG2ALDH1A1GAA
SCHEMBL8433420 0.81 IDH1 (0.42) IDH1ALDH1A1NPC1RAB9AL3MBTL1
Hydrochloric Acid SCHEMBL8434597 0.80 IDH1 (0.41) IDH1ALDH1A1NPC1RAB9AL3MBTL1
Hydrochloric Acid SCHEMBL8495697 0.77 RAB9A (0.44) IDH1LMNANPC1RAB9AL3MBTL1
SCHEMBL8432982 0.75 TAAR1 (0.45) LMNANPC1RAB9AL3MBTL1MEN1
SCHEMBL8438749 0.75 TSHR (0.51) ALDH1A1LMNAL3MBTL1KDM4EMEN1
Hydrochloric Acid SCHEMBL8435752 0.75 TAAR1 (0.44) LMNANPC1RAB9AL3MBTL1MEN1
SCHEMBL8433686 0.74 PTGS1 (0.34) IDH1
SCHEMBL8438545 0.74 SMN1; SMN2 (0.49) ALDH1A1LMNANPC1RAB9AL3MBTL1
Hydrochloric Acid SCHEMBL8437492 0.74 TSHR (0.50) ALDH1A1GAALMNAL3MBTL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5874585-A TREATMENT AND/OR PREVENTION OF ELASTASE-MEDIATED PROBLEMS SUCH AS ARTHRITIS, PERIODONTAL DISEASE, GLOMERULONEPHRITIS, DERMATITIS, PSORIASIS, CYSTIC FIBROSIS, CHRONIC BRONCHITIS, ALZHEIMER'S DISEASE CORTECH, INC. (US) 1999-02-23 US disclosed