SCHEMBL8434278

SCHEMBL8434278

O=C(O)c1ccc(C(=O)c2cc(Cl)cc(Cl)c2)cc1

nearest known ligand 0.72

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 10/20 0.72
TPMT P51580 1/20 0.67
RXRA P19793 2/20 0.64
RXRB P28702 2/20 0.64
TSHR P16473 3/20 0.60
ALOX15 P16050 1/20 0.60
CNR1 P21554 3/20 0.55
CNR2 P34972 3/20 0.55
TP53 P04637 1/20 0.52
HCAR1 Q9BXC0 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11850424 0.86 CNR1 (0.69) SRD5A2TPMTTSHRALOX15CNR1
SCHEMBL9541835 0.84 CNR2 (0.70) SRD5A2TPMTRXRARXRBCNR1
Terephthalic Acid SCHEMBL11195049 0.84 TPMT (0.76) SRD5A2TPMTRXRARXRBTSHR
SCHEMBL4028272 0.84 SRD5A2 (1.00) SRD5A2RXRARXRBTSHRALOX15
SCHEMBL4465360 0.83 TPMT (0.65) SRD5A2TPMTRXRARXRBTSHR
SCHEMBL9360597 0.83 MAPK1 (0.72) SRD5A2TPMTCNR1CNR2HCAR1
SCHEMBL8437706 0.82 SRD5A2 (0.64) SRD5A2RXRARXRBTSHRALOX15
SCHEMBL28565971 0.81 SRD5A2 (0.79) SRD5A2TSHRALOX15TP53
SCHEMBL23699 0.81 TPMT (1.00) SRD5A2TPMTRXRARXRBTSHR
SCHEMBL28214359 0.81 TPMT (1.00) SRD5A2TPMTRXRARXRBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5998433-A THERAPY FOR HYPERLIPIDEMIA; ATHEROSCLEROSIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-12-07 US disclosed
CN-1160403-A Substd. heterobicyclic alkyl amines and their use as squalene oxide cyclase inhibitors TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-09-24 CN disclosed
EP-0785939-A1 SUBSTITUTED HETEROBICYCLIC ALKYL AMINES AND THEIR USE AS SQUALENE OXIDE CYCLASE INHIBITORS Takeda Chemical Industries, Ltd. (JP) 1997-07-30 EP disclosed
WO-1996011201-A1 SUBSTITUTED HETEROBICYCLIC ALKYL AMINES AND THEIR USE AS SQUALENE OXIDE CYCLASE INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-04-18 WO disclosed