SCHEMBL8434406

SCHEMBL8434406

CN(C)Cc1cc2c(o1)CN(C(=O)c1ccc(/C=C\c3ccccc3)cc1)CC2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
HPGD P15428 7/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
TP53 P04637 2/20 0.41
MTHFD1 P11586 1/20 0.40
MTHFD2 P13995 1/20 0.40
LMNA P02545 2/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
SNCA P37840 1/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
RECQL P46063 1/20 0.38
NPSR1 Q6W5P4 2/20 0.38
NPC1 O15118 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPY2R P49146 1/20 0.37
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8436361 1.00 ALDH1A1 (0.41) ALDH1A1HPGDMEN1KMT2ATP53
SCHEMBL8434410 1.00 ALDH1A1 (0.41) ALDH1A1HPGDMEN1KMT2ATP53
Hydrochloric Acid SCHEMBL8440790 0.99 ALDH1A1 (0.41) ALDH1A1HPGDMEN1KMT2ATP53
Hydrochloric Acid SCHEMBL8434573 0.99 ALDH1A1 (0.41) ALDH1A1HPGDMEN1KMT2ATP53
Hydrochloric Acid SCHEMBL8434580 0.99 ALDH1A1 (0.41) ALDH1A1HPGDMEN1KMT2ATP53
SCHEMBL8437896 0.92 LSS (0.44) HPGDKMT2ATP53MTHFD1MTHFD2
SCHEMBL8437891 0.92 LSS (0.44) HPGDKMT2ATP53MTHFD1MTHFD2
SCHEMBL8434898 0.92 ALDH1A1 (0.41) ALDH1A1HPGDMEN1KMT2ATP53
SCHEMBL8434901 0.92 ALDH1A1 (0.41) ALDH1A1HPGDMEN1KMT2ATP53
SCHEMBL8435004 0.92 ALDH1A1 (0.41) ALDH1A1HPGDMEN1KMT2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5998433-A THERAPY FOR HYPERLIPIDEMIA; ATHEROSCLEROSIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-12-07 US disclosed
EP-0785939-A1 SUBSTITUTED HETEROBICYCLIC ALKYL AMINES AND THEIR USE AS SQUALENE OXIDE CYCLASE INHIBITORS Takeda Chemical Industries, Ltd. (JP) 1997-07-30 EP disclosed
WO-1996011201-A1 SUBSTITUTED HETEROBICYCLIC ALKYL AMINES AND THEIR USE AS SQUALENE OXIDE CYCLASE INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-04-18 WO disclosed