SCHEMBL8434648

SCHEMBL8434648

CCCCc1nc(Br)c[nH]1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.46
ALDH1A1 P00352 2/20 0.37
MAPK1 P28482 1/20 0.37
GSK3B P49841 1/20 0.36
PARP1 P09874 1/20 0.36
PKM P14618 1/20 0.35
HPGD P15428 1/20 0.35
GPR84 Q9NQS5 2/20 0.34
HRH4 Q9H3N8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1230952 0.94 ALDH1A1 (0.42) HRH3ALDH1A1PKMHPGDGPR84
SCHEMBL28463361 0.92 ALDH1A1 (0.44) HRH3ALDH1A1PKMHPGDGPR84
Ammonia Solution, Strong SCHEMBL28347379 0.91 ALDH1A1 (0.43) HRH3ALDH1A1PKMHPGDGPR84
SCHEMBL5216842 0.79
SCHEMBL3840247 0.78 HRH3 (0.42) HRH3ALDH1A1MAPK1PARP1PKM
SCHEMBL2037718 0.78 HRH3 (0.42) HRH3ALDH1A1MAPK1PARP1PKM
Hydrochloric Acid SCHEMBL14743464 0.76 HRH3 (0.41) HRH3ALDH1A1MAPK1GSK3BPARP1
SCHEMBL3846855 0.76 HRH3 (0.41) HRH3ALDH1A1MAPK1GSK3BPARP1
SCHEMBL4988560 0.76 HRH3 (0.41) HRH3ALDH1A1MAPK1GSK3BPARP1
SCHEMBL5446824 0.76 HRH3 (0.41) HRH3ALDH1A1MAPK1GSK3BPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021237038-A1 COMPETITIVE AND NONCOMPETITIVE INHIBITORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M5 VANDERBILT UNIVERSITY (US) 2021-11-25 WO disclosed
EP-3438106-A1 ANTI-VIRAL COMPOUNDS AbbVie Ireland Unlimited Company (IE) 2019-02-06 EP disclosed
CN-1238262-C Process for separating and recovering minim organic solvent from waste water using ion liquid INST PROCESS ENG CAS (CN) 2006-01-25 CN disclosed
CN-1594116-A Process for separating and recovering minim organic solvent from waste water using ion liquid INST PROCESS ENG CAS (CN) 2005-03-16 CN disclosed
US-5929249-A ANGIOTENSIN II RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1999-07-27 US disclosed
US-5728842-A ANGIOTENSIN II RECEPTOR ANTAGONIST SMITHKLINE BEECHAM CORPORATION (US) 1998-03-17 US disclosed
EP-0653937-A4 CHEMICAL COMPOUNDS. SMITHKLINE BEECHAM CORP (US) 1996-07-31 EP disclosed
EP-0653937-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1995-05-24 EP disclosed
WO-1994000120-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1994-01-06 WO disclosed