SCHEMBL8436149

SCHEMBL8436149

c1ccc(CNCCc2ccoc2)cc1

nearest known ligand 0.63

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.63
MAPT P10636 1/20 0.63
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
TDP1 Q9NUW8 1/20 0.55
SIGMAR1 Q99720 3/20 0.50
MAOA P21397 1/20 0.50
BCHE P06276 2/20 0.49
MPO P05164 2/20 0.49
CHRM2 P08172 1/20 0.48
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA4 P22748 1/20 0.47
CA9 Q16790 1/20 0.47
ATM Q13315 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6421867 0.85 MEN1 (0.52) GAAMAPTMEN1KMT2ATDP1
SCHEMBL27228 0.80 GAA (0.95) GAAMAPTMEN1KMT2ATDP1
SCHEMBL8439993 0.80 SIGMAR1 (0.70) SIGMAR1MAOABCHECHRM2
Hydrochloric Acid SCHEMBL1983401 0.78 GAA (1.00) GAAMAPTMEN1KMT2ATDP1
SCHEMBL11881258 0.78 GAA (0.91) GAAMAPTMEN1KMT2ATDP1
Ammonia Solution, Strong SCHEMBL23581968 0.78 GAA (0.91) GAAMAPTMEN1KMT2ATDP1
SCHEMBL25432637 0.78 GAA (0.91) GAAMAPTMEN1KMT2ATDP1
SCHEMBL3272134 0.78 GAA (0.91) GAAMAPTMEN1KMT2ATDP1
SCHEMBL5069114 0.76 CA1 (0.51) GAAMAPTSIGMAR1BCHEKDM4E
SCHEMBL11877395 0.75 GAA (0.76) GAAMAPTMEN1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5998433-A THERAPY FOR HYPERLIPIDEMIA; ATHEROSCLEROSIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-12-07 US disclosed
CN-1160403-A Substd. heterobicyclic alkyl amines and their use as squalene oxide cyclase inhibitors TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-09-24 CN disclosed
EP-0785939-A1 SUBSTITUTED HETEROBICYCLIC ALKYL AMINES AND THEIR USE AS SQUALENE OXIDE CYCLASE INHIBITORS Takeda Chemical Industries, Ltd. (JP) 1997-07-30 EP disclosed
WO-1996011201-A1 SUBSTITUTED HETEROBICYCLIC ALKYL AMINES AND THEIR USE AS SQUALENE OXIDE CYCLASE INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-04-18 WO disclosed