SCHEMBL8437222

SCHEMBL8437222

CN(C)Cc1cc2c(o1)CCN(C(=O)c1ccc(C(=O)c3ccccc3)cc1)CC2

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.47
POLB P06746 1/20 0.43
ALDH1A1 P00352 4/20 0.42
ACHE P22303 1/20 0.40
SLC6A7 Q99884 1/20 0.40
LSS P48449 1/20 0.40
CYP2C9 P11712 1/20 0.40
PLA2G1B P04054 1/20 0.40
ATG4B Q9Y4P1 1/20 0.40
MTHFD1 P11586 1/20 0.40
MTHFD2 P13995 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
BLM P54132 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8437586 0.99 HPGD (0.46) HPGDPOLBALDH1A1ACHESLC6A7
SCHEMBL8439848 0.93 ALDH1A1 (0.43) HPGDPOLBALDH1A1PLA2G1BATG4B
SCHEMBL8439061 0.93 ALDH1A1 (0.43) HPGDPOLBALDH1A1MTHFD1MTHFD2
Hydrochloric Acid SCHEMBL8436197 0.92 ALDH1A1 (0.43) HPGDPOLBALDH1A1MTHFD1MTHFD2
Hydrochloric Acid SCHEMBL8439685 0.92 ALDH1A1 (0.43) HPGDPOLBALDH1A1PLA2G1BATG4B
Hydrochloric Acid SCHEMBL8804440 0.92 ALDH1A1 (0.43) HPGDPOLBALDH1A1PLA2G1BATG4B
SCHEMBL27464735 0.88 ALDH1A1 (0.44) HPGDALDH1A1CYP2C9MTHFD1MTHFD2
SCHEMBL8436364 0.86 ALDH1A1 (0.42) HPGDALDH1A1MTHFD1MTHFD2
SCHEMBL8434934 0.86 HDAC6 (0.42) HPGDPOLBALDH1A1PLA2G1BATG4B
SCHEMBL8436047 0.86 HPGD (0.42) HPGDALDH1A1MTHFD1MTHFD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5998433-A THERAPY FOR HYPERLIPIDEMIA; ATHEROSCLEROSIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-12-07 US disclosed
CN-1160403-A Substd. heterobicyclic alkyl amines and their use as squalene oxide cyclase inhibitors TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-09-24 CN disclosed
EP-0785939-A1 SUBSTITUTED HETEROBICYCLIC ALKYL AMINES AND THEIR USE AS SQUALENE OXIDE CYCLASE INHIBITORS Takeda Chemical Industries, Ltd. (JP) 1997-07-30 EP disclosed
WO-1996011201-A1 SUBSTITUTED HETEROBICYCLIC ALKYL AMINES AND THEIR USE AS SQUALENE OXIDE CYCLASE INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-04-18 WO disclosed