SCHEMBL8437671

SCHEMBL8437671

O=C(O)c1ccc(C(=O)c2ccco2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.68
MEN1 O00255 1/20 0.68
POLB P06746 1/20 0.68
THRB P10828 1/20 0.68
APEX1 P27695 1/20 0.68
RECQL P46063 1/20 0.68
KMT2A Q03164 1/20 0.68
TDP1 Q9NUW8 1/20 0.68
SRD5A2 P31213 6/20 0.54
CES2 O00748 1/20 0.54
CES1 P23141 1/20 0.54
PTPN1 P18031 1/20 0.53
TSHR P16473 2/20 0.50
CSNK2A2 P19784 1/20 0.49
CSNK2A1 P68400 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
TP53 P04637 1/20 0.48
RAB9A P51151 2/20 0.46
BLM P54132 1/20 0.46
PIM1 P11309 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3953437 0.88 ALDH1A1 (0.73) ALDH1A1MEN1POLBTHRBAPEX1
SCHEMBL29029980 0.86 KMT2A (0.85) ALDH1A1MEN1POLBTHRBAPEX1
SCHEMBL459833 0.84 MEN1 (0.68) ALDH1A1MEN1POLBTHRBAPEX1
SCHEMBL10682751 0.82 ALDH1A1 (0.66) ALDH1A1MEN1POLBTHRBAPEX1
SCHEMBL16713290 0.82 KMT2A (0.66) ALDH1A1MEN1POLBTHRBAPEX1
SCHEMBL11112092 0.82 KMT2A (0.66) ALDH1A1MEN1POLBTHRBAPEX1
SCHEMBL11616485 0.82 ALDH1A1 (0.62) ALDH1A1MEN1POLBTHRBAPEX1
SCHEMBL15354269 0.81 ALDH1A1 (1.00) ALDH1A1MEN1POLBTHRBAPEX1
SCHEMBL13052375 0.80 ALDH1A1 (0.58) ALDH1A1MEN1POLBTHRBAPEX1
SCHEMBL25498872 0.80 ALDH1A1 (0.58) ALDH1A1MEN1POLBTHRBAPEX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12509465-B2 Benzoimidazole derivatives as anticancer agents CENTRE LEON BERARD (FR) 2025-12-30 US disclosed
EP-3515904-B1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS CENTRE LEON BERARD (FR) 2024-01-17 EP disclosed
CN-110234640-B Benzimidazole derivatives as anticancer agents 利昂贝拉尔中心 2023-04-07 CN disclosed
US-20220348587-A1 Benzoimidazole Derivatives As Anticancer Agents CENTRE LEON BERARD (FR) 2022-11-03 US disclosed
US-11384081-B2 Benzoimidazole derivatives as anticancer agents CENTRE LEON BERARD (FR) 2022-07-12 US disclosed
US-20210292328-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS CENTRE LEON BERARD (FR) 2021-09-23 US disclosed
CN-110234640-A Benzimidazole derivatives as anticancer agents 利昂贝拉尔中心 2019-09-13 CN disclosed
EP-3515904-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS Centre Leon Berard (FR) 2019-07-31 EP disclosed
WO-2018054989-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS CENTRE LEON BERARD (FR) 2018-03-29 WO disclosed
US-5998433-A THERAPY FOR HYPERLIPIDEMIA; ATHEROSCLEROSIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-12-07 US disclosed
CN-1160403-A Substd. heterobicyclic alkyl amines and their use as squalene oxide cyclase inhibitors TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-09-24 CN disclosed
EP-0785939-A1 SUBSTITUTED HETEROBICYCLIC ALKYL AMINES AND THEIR USE AS SQUALENE OXIDE CYCLASE INHIBITORS Takeda Chemical Industries, Ltd. (JP) 1997-07-30 EP disclosed
WO-1996011201-A1 SUBSTITUTED HETEROBICYCLIC ALKYL AMINES AND THEIR USE AS SQUALENE OXIDE CYCLASE INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-04-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12509465-B2 Benzoimidazole derivatives as anticancer agents CCAR2, MAPKAP1, BCOR ALDH1A1 3500/4885MEN1 4170/4885POLB 2146/4885
US-20210292328-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS TMBIM6, BAX, MAPK14 ALDH1A1 2866/4885MEN1 4272/4885POLB 1598/4885
US-11384081-B2 Benzoimidazole derivatives as anticancer agents TMBIM6, BAX, MAPK14 ALDH1A1 2866/4885MEN1 4272/4885POLB 1598/4885
US-20220348587-A1 Benzoimidazole Derivatives As Anticancer Agents TMBIM6, BAX, BCL2 ALDH1A1 2871/4885MEN1 4350/4885POLB 1569/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.