SCHEMBL8438398

SCHEMBL8438398

FC(F)(F)c1cncc(OC[C@@H]2CCN2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 4/20 0.64
CHRNA4 P43681 3/20 0.64
KDM4E B2RXH2 1/20 0.63
CYP1A2 P05177 1/20 0.63
CYP2D6 P10635 1/20 0.63
CYP2C9 P11712 1/20 0.63
CYP2C19 P33261 1/20 0.63
CHRNA6 Q15825 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8437910 0.99 CHRNB2 (0.63) CHRNB2CHRNA4KDM4ECYP1A2CYP2D6
SCHEMBL8435051 0.91 CHRNB4 (0.66) CHRNB2CHRNA4
SCHEMBL8440255 0.91 CHRNB4 (0.66) CHRNB2CHRNA4
Hydrochloric Acid SCHEMBL7455989 0.89 CHRNB4 (0.64) CHRNB2CHRNA4
Hydrochloric Acid SCHEMBL7411399 0.89 CHRNB4 (0.64) CHRNB2CHRNA4
SCHEMBL4111623 0.81 CHRNB2 (0.68) CHRNB2CHRNA4KDM4ECYP1A2CYP2D6
SCHEMBL7411369 0.81 CHRNB2 (0.68) CHRNB2CHRNA4KDM4ECYP1A2CYP2D6
SCHEMBL12557242 0.81 CHRNB2 (0.68) CHRNB2CHRNA4KDM4ECYP1A2CYP2D6
Hydrochloric Acid SCHEMBL30785448 0.81 KDM1A (0.53) CHRNB2CHRNA4CHRNA6
Hydrochloric Acid SCHEMBL27159065 0.81 KDM1A (0.53) CHRNB2CHRNA4CHRNA6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5914328-A CONTROL DOPAMINE RELEASE, ACTIVATE CHOLINERGIC CHANNELS ABBOTT LABORATORIES (US) 1999-06-22 US claimed
US-5914328-A CONTROL DOPAMINE RELEASE, ACTIVATE CHOLINERGIC CHANNELS ABBOTT LABORATORIES (US) 1999-06-22 US disclosed