SCHEMBL8438403

SCHEMBL8438403

O=[N+]([O-])c1ccc(N2CCC(O)C(N3CCC(c4ccccc4)CC3)C2)cc1

nearest known ligand 0.98

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC18A3 Q16572 8/20 0.62
CYP2D6 P10635 2/20 0.51
TSHR P16473 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
SIGMAR1 Q99720 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2C9 P11712 1/20 0.51
ALDH1A1 P00352 1/20 0.50
APEX1 P27695 1/20 0.50
BLM P54132 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6714666 0.83 MAPT (0.53) SMN1; SMN2CYP2C9ALDH1A1
SCHEMBL242050 0.83 MAPT (0.59) SLC18A3SMN1; SMN2CYP2C9ALDH1A1
SCHEMBL7301802 0.81 TRPV6 (0.59) SLC18A3CYP2D6CYP2C9ALDH1A1
SCHEMBL6610401 0.77 MEN1 (0.59) SMN1; SMN2CYP2C9ALDH1A1
SCHEMBL31224897 0.76 MAPT (0.55) CYP2C9ALDH1A1
SCHEMBL7300130 0.75 MAPT (0.55) SMN1; SMN2CYP2C9ALDH1A1
SCHEMBL31224958 0.75 MAPT (0.51) SMN1; SMN2CYP2C9ALDH1A1
SCHEMBL9984902 0.73 POLB (0.51) CYP2C9ALDH1A1
SCHEMBL854301 0.72 MAPT (0.56) CYP2C9ALDH1A1
SCHEMBL2126184 0.72 MAPT (0.56) CYP2C9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5876694-A NON-INVASIVELY MAPPING CHOLINERGIC INNERVATION IN A LIVING BRAIN COMPRISES INJECTING THE BRAIN WITH A RADIOLABELLED VESAMICOL DERIVATIVE, MAGNETIC RESONANCE IMAGING REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 1999-03-02 US disclosed
US-5789420-A Azavesamicols REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 1998-08-04 US disclosed
EP-0643696-A1 AZAVESAMICOLS THE REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 1995-03-22 EP disclosed
EP-0643696-A4 AZAVESAMICOLS. UNIV MINNESOTA (US) 1995-01-20 EP disclosed
US-5338852-A Azavesamicols REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 1994-08-16 US disclosed
WO-1993024457-A1 AZAVESAMICOLS REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 1993-12-09 WO disclosed