SCHEMBL8439844

SCHEMBL8439844

CN(C(=O)OCc1ccc([N+](=O)[O-])cc1)N1CC[C@H](OC(=O)C(F)(F)F)C1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.40
CCR5 P51681 10/20 0.40
TDP1 Q9NUW8 1/20 0.39
ALDH1A1 P00352 2/20 0.39
KCNJ1 P48048 1/20 0.39
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
BCHE P06276 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8095172 0.76 CCR5 (0.42) CCR5
SCHEMBL7732703 0.71 CCR5 (0.53) CCR5
SCHEMBL994551 0.71 MAPT (0.40) ATMTDP1ALDH1A1MAPTHPGD
SCHEMBL994549 0.71 MAPT (0.40) ATMTDP1ALDH1A1MAPTHPGD
SCHEMBL6767786 0.70 KDM4E (0.43) ATMCCR5TDP1ALDH1A1MAPT
SCHEMBL5724304 0.70 ALDH1A1 (0.47) TDP1ALDH1A1MAPTHPGDBCHE
SCHEMBL10639614 0.70 SMN1; SMN2 (0.47) TDP1ALDH1A1MAPTHPGD
Trifluoroacetic Acid SCHEMBL8095167 0.69 SLC6A2 (0.41) CCR5ALDH1A1KCNJ1
SCHEMBL8439868 0.68 EPHX1 (0.45) TDP1KCNJ1
SCHEMBL8438723 0.68 EPHX1 (0.45) TDP1KCNJ1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5866564-A STABILITY SANKYO COMPANY, LIMITED (JP) 1999-02-02 US disclosed
US-5712267-A Carbapenem derivatives, their preparation and their use as antibiotics SANKYO COMPANY,. LIMITED (JP) 1998-01-27 US disclosed