SCHEMBL8440267

SCHEMBL8440267

CCN(CC)CCNC(=O)c1cc(C(=O)OC)cc(-c2cc(Cl)sc2Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
ALDH1A1 P00352 5/20 0.42
LMNA P02545 4/20 0.42
SLC22A1 O15245 2/20 0.42
KCNH2 Q12809 2/20 0.42
HTR3E A5X5Y0 1/20 0.42
HTR3B O95264 1/20 0.42
MPO P05164 1/20 0.42
CYP1A2 P05177 1/20 0.42
ADRA2A P08913 1/20 0.42
CYP2D6 P10635 1/20 0.42
DRD2 P14416 1/20 0.42
ADRA2C P18825 1/20 0.42
DRD4 P21917 1/20 0.42
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
DRD3 P35462 1/20 0.42
HTR2B P41595 1/20 0.42
HTR3A P46098 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8440805 0.94 MAPK1 (0.42) TMEM97SIGMAR1ALDH1A1LMNATSHR
SCHEMBL8440765 0.89 MAPK1 (0.45) ALDH1A1LMNACYP1A2MAPK1SMN1; SMN2
SCHEMBL8439277 0.85 PDE4B (0.43) TMEM97SIGMAR1ALDH1A1MAPK1RAB9A
SCHEMBL8444315 0.81 CA12 (0.42) ALDH1A1LMNARAB9ANFKB1SMN1; SMN2
SCHEMBL7995581 0.81 MCHR1 (0.46) TMEM97SIGMAR1ALDH1A1LMNASLC22A1
Hydrochloric Acid SCHEMBL8817606 0.79 HRH3 (0.40) CYP2D6ACHEPMP22CYP3A4SMN1; SMN2
Hydrochloric Acid SCHEMBL8440407 0.78 SMN1; SMN2 (0.52) ALDH1A1LMNAHTR4SMN1; SMN2POLB
Hydrochloric Acid SCHEMBL8440293 0.78 APP (0.53) ALDH1A1LMNACYP1A2CYP2D6HTR4
SCHEMBL8440888 0.77 LMNA (0.53) ALDH1A1LMNAKCNH2CYP1A2CYP2D6
SCHEMBL8441395 0.76 DAO (0.40) ALDH1A1LMNATSHRRAB9ANFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5968985-A INHIBITORS OF SODIUM ION/HYDROGEN ION EXCHANGE IN CELLS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-10-19 US disclosed
EP-0773927-A2 BENZOYLGUANIDINE DERIVATIVES AS MEDICAMENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-05-21 EP disclosed
WO-1996004241-A2 BENZOYLGUANIDINE DERIVATIVES AS MEDICAMENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-02-15 WO disclosed