SCHEMBL8440317

SCHEMBL8440317

Clc1ccc(CCBr)c(Cl)c1Cl

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.39
CYP3A4 P08684 1/20 0.37
MAPK1 P28482 1/20 0.37
AHR P35869 2/20 0.37
PNMT P11086 1/20 0.33
TDP1 Q9NUW8 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11311694 0.80 MEP1A (0.34) TAAR1CYP3A4MAPK1
SCHEMBL6305999 0.80 CYP3A4 (0.40) TAAR1CYP3A4MAPK1AHRPNMT
SCHEMBL3124138 0.79 TAAR1 (0.63) TAAR1CYP3A4PNMT
SCHEMBL30252677 0.79 TAAR1 (0.63) TAAR1CYP3A4PNMT
SCHEMBL10920592 0.79 TAAR1 (0.31) TAAR1
SCHEMBL9482589 0.78 TAAR1 (0.40) TAAR1CYP3A4MAPK1AHRPNMT
SCHEMBL8893652 0.76 TAAR1 (0.65) TAAR1CYP3A4MAPK1PNMT
SCHEMBL10061111 0.76 TAAR1 (0.39) TAAR1CYP3A4MAPK1AHRPNMT
SCHEMBL17552721 0.76 TAAR1 (0.39) TAAR1CYP3A4MAPK1AHRPNMT
SCHEMBL5477243 0.76

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0604857-B1 Process for preparing optically active 4-mercapto-2-pyrrolidone derivative and intermediate therefor TANABE SEIYAKU CO (JP) 1999-03-17 EP disclosed
US-5495012-A Process for preparing optically active 4-mercapto-2-pyrrolidone derivative and intermediate therefor TANABE SEIYAKU CO., LTD. (JP) 1996-02-27 US disclosed
US-5424446-A Process for preparing optically active 4-mercapto-2-pyrrolidone derivative and intermediate therefor TANABE SEIYAKU CO., LTD. (JP) 1995-06-13 US disclosed
EP-0604857-A1 Process for preparing optically active 4-mercapto-2-pyrrolidone derivative and intermediate therefor TANABE SEIYAKU CO., LTD. (JP) 1994-07-06 EP disclosed