SCHEMBL8440353

SCHEMBL8440353

Cc1c(Cc2ccccc2)ccc2c(O)cc(=O)oc12

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.57
CNR2 P34972 3/20 0.56
GPR55 Q9Y2T6 3/20 0.56
SHBG P04278 1/20 0.53
MAOB P27338 1/20 0.52
CA12 O43570 2/20 0.52
CA9 Q16790 2/20 0.52
HSD17B3 P37058 2/20 0.52
TNF P01375 1/20 0.52
NOD2 Q9HC29 1/20 0.52
NOD1 Q9Y239 1/20 0.52
GAA P10253 3/20 0.50
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
ALDH1A1 P00352 2/20 0.50
GLA P06280 2/20 0.50
HPGD P15428 1/20 0.50
TSHR P16473 1/20 0.50
CASP1 P29466 1/20 0.50
CASP7 P55210 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8441390 0.82 KDM4E (0.63) KDM4EMAOBCA9ALDH1A1HPGD
SCHEMBL19019865 0.79 KDM4E (0.53) KDM4ECA12CA9TNFNOD2
SCHEMBL5345045 0.77 MAOB (0.77) KDM4EMAOBCA12CA9TNF
SCHEMBL5346589 0.76 MAOB (0.65) KDM4EMAOBCA12CA9TNF
SCHEMBL8442563 0.74 HPGD (0.72) KDM4EMAOBGAAMEN1KMT2A
SCHEMBL2761835 0.72 MET (0.56) KDM4EMAOBCA12CA9TNF
SCHEMBL19019871 0.72 KDM4E (0.51) KDM4ECA12CA9TNFNOD2
SCHEMBL19019924 0.72 TDP1 (0.53) KDM4EMAOBCA12CA9MAOA
SCHEMBL19275311 0.72 GPR55 (0.46) KDM4ECNR2GPR55SHBGALDH1A1
SCHEMBL3575287 0.72 MET (0.56) KDM4EMAOBCA12CA9TNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5985912-A COUMARONE COMPOUNDS AS BACTERICIDES PFIZER INC. (US) 1999-11-16 US disclosed
US-5624951-A 4-hydroxy coumarin derivatives with antibacterial activity PFIZER INC. (US) 1997-04-29 US disclosed
EP-0658158-A1 4-HYDROXY COUMARIN DERIVATIVES WITH ANTIBACTERIAL ACTIVITY PFIZER INC. (US) 1995-06-21 EP disclosed
WO-1994005649-A1 4-HYDROXY COUMARIN DERIVATIVES WITH ANTIBACTERIAL ACTIVITY PFIZER INC. (US) 1994-03-17 WO disclosed