SCHEMBL8440981

SCHEMBL8440981

COC(=O)c1cccc(-c2c(Cl)cccc2Cl)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.52
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
CA9 Q16790 1/20 0.52
NR1H2 P55055 1/20 0.52
NR1H3 Q13133 1/20 0.52
MAPT P10636 4/20 0.51
ERN1 O75460 3/20 0.51
NPC1 O15118 3/20 0.51
RAB9A P51151 3/20 0.51
KMT2A Q03164 2/20 0.51
MEN1 O00255 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
NR1H4 Q96RI1 1/20 0.49
ALDH1A1 P00352 2/20 0.49
POLB P06746 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28409132 0.84 ERN1 (0.50) CA12CA1CA2CA9NR1H2
SCHEMBL3316502 0.84 CYP19A1 (0.56) NR1H2NR1H3ERN1ALDH1A1PLAU
SCHEMBL7844717 0.84 KAT6A (0.53) CA12CA1CA2CA9MAPT
SCHEMBL67941 0.84 CA12 (0.68) CA12CA1CA2CA9ERN1
SCHEMBL8444016 0.83 RXRA (0.65) CA12CA1CA2CA9MAPT
SCHEMBL2035024 0.83 TSHR (0.52) CA12CA1CA2CA9MAPT
SCHEMBL8443917 0.83 KMT2A (0.52) CA12CA1CA2CA9MAPT
SCHEMBL27715902 0.82 CA12 (0.71) CA12CA1CA2CA9ERN1
SCHEMBL7827008 0.81 PLAU (0.59) CA12CA1CA2CA9MAPT
SCHEMBL5423712 0.80 HDAC8 (0.54) NR1H2NR1H3ALDH1A1POLBCDK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5968985-A INHIBITORS OF SODIUM ION/HYDROGEN ION EXCHANGE IN CELLS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-10-19 US disclosed
EP-0773927-A2 BENZOYLGUANIDINE DERIVATIVES AS MEDICAMENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-05-21 EP disclosed
WO-1996004241-A2 BENZOYLGUANIDINE DERIVATIVES AS MEDICAMENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-02-15 WO disclosed