SCHEMBL8442174

SCHEMBL8442174

COc1ccccc1N1CCN(CC(c2ccccc2)C2(C(=O)O)CCCCC2)CC1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 5/20 0.57
ALDH1A1 P00352 3/20 0.57
KDM4E B2RXH2 2/20 0.57
CYP1A2 P05177 1/20 0.57
CYP3A4 P08684 1/20 0.57
CYP2D6 P10635 1/20 0.57
ALOX15 P16050 1/20 0.57
HSD17B10 Q99714 1/20 0.57
HTR1D P28221 1/20 0.56
HTR2B P41595 1/20 0.56
LMNA P02545 1/20 0.52
ADRA1B P35368 3/20 0.51
TDP1 Q9NUW8 1/20 0.51
IGF1R P08069 1/20 0.51
ADRB2 P07550 1/20 0.49
ADRB1 P08588 1/20 0.49
ADRB3 P13945 1/20 0.49
ADRA1D P25100 1/20 0.49
ADRA1A P35348 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8442538 0.78 HTR1A (0.76) HTR1AALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL9004457 0.78 HTR1A (0.80) HTR1AALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL8442654 0.78 HTR1A (0.80) HTR1AALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL8442467 0.77 HTR1A (0.78) HTR1AALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL8442968 0.76 HTR1A (0.78) HTR1AALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL8444529 0.76 HTR1A (0.75) HTR1AALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL8442587 0.76 IGF1R (0.81) HTR1AALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL7699947 0.76 ALDH1A1 (0.46) HTR1AALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL8443682 0.76 HTR1A (0.72) HTR1AALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL7777456 0.76 HTR1A (0.63) HTR1AALDH1A1KDM4ECYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0395312-B1 Piperazine derivatives WYETH JOHN & BROTHER LTD (GB) 1999-05-12 EP claimed