SCHEMBL8443151

SCHEMBL8443151

CCOc1cc(C(=O)OC)c(OC2CCCCO2)c(NS(=O)(=O)c2ccc(OC)cc2)c1Oc1cc(OC)ccc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.41
MAPT P10636 4/20 0.41
EDNRA P25101 1/20 0.40
LMNA P02545 7/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
HTT P42858 4/20 0.37
MAPK1 P28482 1/20 0.37
KDM4E B2RXH2 3/20 0.37
RCE1 Q9Y256 1/20 0.37
HPGD P15428 2/20 0.37
HSD17B10 Q99714 1/20 0.37
KMT2A Q03164 3/20 0.36
MEN1 O00255 1/20 0.36
GAA P10253 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
NPC1 O15118 2/20 0.36
TSHR P16473 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
TP53 P04637 2/20 0.36
USP2 O75604 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8441685 0.95 EDNRA (0.46) ALDH1A1MAPTEDNRALMNASMN1; SMN2
SCHEMBL8445360 0.94 ALDH1A1 (0.42) ALDH1A1MAPTEDNRALMNASMN1; SMN2
SCHEMBL8441557 0.90 ALDH1A1 (0.42) ALDH1A1MAPTEDNRALMNASMN1; SMN2
SCHEMBL8445338 0.90 ALDH1A1 (0.41) ALDH1A1MAPTEDNRALMNASMN1; SMN2
SCHEMBL8443878 0.87 EDNRA (0.36) EDNRANPC1RAB9A
SCHEMBL8445329 0.86 NPC1 (0.38) ALDH1A1MAPTLMNAKDM4EHSD17B10
SCHEMBL8441255 0.85 EDNRA (0.40) ALDH1A1MAPTEDNRALMNASMN1; SMN2
SCHEMBL8444402 0.84 NPC1 (0.37) ALDH1A1MAPTEDNRALMNASMN1; SMN2
SCHEMBL8444252 0.84 EDNRB (0.46) EDNRA
SCHEMBL8445313 0.84 EDNRB (0.44) ALDH1A1MAPTEDNRALMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5962682-A Aryl- and hetaryl-sulfonamide derivatives, their preparation and their use as endothelin antagonists HOFFMANN-LA ROCHE INC. (US) 1999-10-05 US disclosed