SCHEMBL8444402

SCHEMBL8444402

CCOc1cc(C(=O)OC)c(OC2CCCCO2)c([N+](=O)[O-])c1Oc1cc(OC)ccc1Cl

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.37
RAB9A P51151 5/20 0.37
POLB P06746 1/20 0.35
CREBBP Q92793 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
TDP1 Q9NUW8 3/20 0.33
ALDH1A1 P00352 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
KMT2A Q03164 2/20 0.33
LMNA P02545 2/20 0.33
EDNRA P25101 1/20 0.33
MAPT P10636 2/20 0.33
MEN1 O00255 1/20 0.33
ALOX12 P18054 1/20 0.33
CASP3 P42574 1/20 0.33
SENP7 Q9BQF6 1/20 0.33
KDM4E B2RXH2 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8444952 0.88 LMNA (0.37) NPC1RAB9APOLBCREBBPTDP1
SCHEMBL8445329 0.88 NPC1 (0.38) NPC1RAB9APOLBCREBBPPTGDR2
SCHEMBL8445321 0.87 CREBBP (0.36) NPC1RAB9ACREBBPTDP1ALDH1A1
SCHEMBL8443151 0.84 ALDH1A1 (0.41) NPC1RAB9APOLBALDH1A1SMN1; SMN2
SCHEMBL8442125 0.84 CREBBP (0.38) POLBCREBBPTDP1ALDH1A1SMN1; SMN2
SCHEMBL8441685 0.82 EDNRA (0.46) ALDH1A1SMN1; SMN2KMT2ALMNAEDNRA
SCHEMBL8445360 0.79 ALDH1A1 (0.42) NPC1TDP1ALDH1A1SMN1; SMN2KMT2A
SCHEMBL8443878 0.78 EDNRA (0.36) NPC1RAB9AEDNRA
SCHEMBL8441255 0.77 EDNRA (0.40) ALDH1A1SMN1; SMN2KMT2ALMNAEDNRA
SCHEMBL7569402 0.76 HPGD (0.39) NPC1RAB9APOLBALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5962682-A Aryl- and hetaryl-sulfonamide derivatives, their preparation and their use as endothelin antagonists HOFFMANN-LA ROCHE INC. (US) 1999-10-05 US disclosed