SCHEMBL8443280

SCHEMBL8443280

O=C(O)c1cccc(-c2coc3ccccc23)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.53
KEAP1 Q14145 1/20 0.49
NPC1 O15118 1/20 0.47
POLB P06746 1/20 0.47
MAPK1 P28482 1/20 0.47
MAP2K4 P45985 1/20 0.47
MAPKAPK3 Q16644 1/20 0.47
MAPK6 Q16659 1/20 0.47
MIF P14174 1/20 0.47
MAOB P27338 1/20 0.46
AXL P30530 1/20 0.45
RXRA P19793 1/20 0.44
RXRB P28702 1/20 0.44
PTPN1 P18031 1/20 0.44
DDT P30046 1/20 0.43
TTR P02766 2/20 0.43
GSK3B P49841 1/20 0.43
PTGER1 P34995 1/20 0.43
FOLH1 Q04609 1/20 0.43
PIN1 Q13526 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11550173 0.83 GSK3B (0.51) KMOKEAP1NPC1POLBMAOB
SCHEMBL8443258 0.83 AXL (0.49) NPC1POLBAXLGSK3BPIN1
SCHEMBL11550178 0.83 SMN1; SMN2 (0.48) KMOKEAP1NPC1POLBRXRA
SCHEMBL11458495 0.83 GSK3B (0.56) NPC1POLBMAP2K4MIFMAOB
SCHEMBL8802708 0.82 KEAP1 (0.53) KMOKEAP1POLBAXLRXRA
SCHEMBL11623160 0.81 PIN1 (0.55) KMONPC1POLBMAPK1TTR
SCHEMBL11620715 0.81 POLB (0.59) KMONPC1POLBTTRGSK3B
SCHEMBL21310963 0.78 KDM4C (0.54) KMOMAOBIKBKETBK1
SCHEMBL23972419 0.78 PLA2G10 (0.48) NPC1POLBMIF
SCHEMBL1310425 0.78 PIN1 (0.56) NPC1POLBMAPK1MIFMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113321640-B Indole compound and application thereof 中国科学院广州生物医药与健康研究院 2023-06-09 CN disclosed
CN-109111427-B Indole compound and application thereof 中国科学院广州生物医药与健康研究院 2023-06-02 CN disclosed
US-5968985-A INHIBITORS OF SODIUM ION/HYDROGEN ION EXCHANGE IN CELLS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-10-19 US disclosed
EP-0773927-A2 BENZOYLGUANIDINE DERIVATIVES AS MEDICAMENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-05-21 EP disclosed
WO-1996004241-A2 BENZOYLGUANIDINE DERIVATIVES AS MEDICAMENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-02-15 WO disclosed
US-4212865-A BACTERICIDES RIKER LABORATORIES, INC. (US) 1980-07-15 US disclosed
US-4190590-A DISINFECTING AND STERILIZING DENTAL AND MEDICAL EQUIPMENT RIKER LABORATORIES, INC. (US) 1980-02-26 US disclosed
US-4124602-A OPTIONALLY SUBSTITUTED 3-(CYANOPHENYL)BENZOFURANS RIKER LABORATORIES, INC. (US) 1978-11-07 US disclosed
US-4048323-A Antimicrobial (2-nitro-3-benzofuranyl)-benzoic acids RIKER LABORATORIES, INC. (US) 1977-09-13 US disclosed