SCHEMBL8445007

SCHEMBL8445007

Bc1cn(S(=O)(=O)c2ccccc2)c2ncc(N3C(=O)c4ccccc4C3=O)cc12

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.39
LMNA P02545 1/20 0.39
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
CA12 O43570 2/20 0.37
CA9 Q16790 2/20 0.37
SCN2A Q99250 1/20 0.37
HTR6 P50406 6/20 0.35
HTT P42858 1/20 0.35
RXFP1 Q9HBX9 2/20 0.35
DRD2 P14416 2/20 0.35
HTR2A P28223 2/20 0.35
HTR1A P08908 1/20 0.35
HTR7 P34969 1/20 0.35
CYP2C19 P33261 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3348657 0.86 CA1 (0.40) BRD4LMNACA1CA2CA12
SCHEMBL16884156 0.70 PTPN11 (0.41) BRD4LMNACA1CA2HTT
SCHEMBL8443828 0.68 MEN1 (0.40) CA1CA2CA12CA9SCN2A
SCHEMBL13505081 0.68 KMT2A (0.47) BRD4HTTRXFP1KMT2A
SCHEMBL13505057 0.67 KMT2A (0.39) CA1CA2CA12CA9SCN2A
SCHEMBL8298982 0.67 BRD4 (0.41) BRD4HTR6DRD2HTR2AHTR1A
SCHEMBL14049066 0.67 BRD4 (0.39) BRD4CA1CA2CA12CA9
SCHEMBL13620691 0.66 HTR6 (0.53) BRD4CA1CA2CA12CA9
SCHEMBL8192188 0.65 PDPK1 (0.47) BRD4CA1CA2CA12CA9
SCHEMBL12657360 0.65 L3MBTL1 (0.58) HTR6HTTCYP2C19KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1749829-B1 JNK inhibitors EISAI R&D MAN CO LTD (JP) 2010-11-03 EP disclosed
EP-1749829-A1 JNK inhibitors Eisai London Research Laboratories Limited (GB) 2007-02-07 EP disclosed