SCHEMBL8445530

SCHEMBL8445530

NS(=O)(=O)c1c(Cc2ccc3c(c2)OCO3)sc2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.46
HSD17B10 Q99714 1/20 0.46
VKORC1 Q9BQB6 1/20 0.42
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
HPGD P15428 3/20 0.42
KDM4E B2RXH2 2/20 0.42
MAPT P10636 2/20 0.42
GAA P10253 2/20 0.42
POLB P06746 1/20 0.42
LMNA P02545 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HTT P42858 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
USP2 O75604 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
HSP90AB1 P08238 2/20 0.39
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6956724 0.88 ALDH1A1 (0.43) ALDH1A1HSD17B10VKORC1MEN1KMT2A
SCHEMBL7212878 0.77 EDNRA (0.53) ALDH1A1HSD17B10MEN1KMT2AHPGD
SCHEMBL4630726 0.76 EDNRA (0.47) ALDH1A1HSD17B10MEN1KMT2AHPGD
SCHEMBL6150865 0.75 EDNRA (0.54)
SCHEMBL4630675 0.75 EDNRB (0.58)
SCHEMBL7977965 0.73 PTGS1 (0.42) ALDH1A1HSD17B10MEN1KMT2AHPGD
SCHEMBL8915088 0.72 EDNRB (0.55)
SCHEMBL15647892 0.71 TAAR1 (0.45) ALDH1A1VKORC1MEN1KMT2AHTT
SCHEMBL7343886 0.70 CNR2 (0.43) ALDH1A1MAPTL3MBTL1
SCHEMBL6968498 0.68 ALDH1A1 (0.48) ALDH1A1HSD17B10MEN1KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946552-A1 SULFONAMIDES AND DERIVATIVES THEREOF THAT MODULATE THE ACTIVITY OF ENDOTHELIN TEXAS BIOTECHNOLOGY CORPORATION (US) 1999-10-06 EP disclosed
WO-1998013366-A1 SULFONAMIDES AND DERIVATIVES THEREOF THAT MODULATE THE ACTIVITY OF ENDOTHELIN TEXAS BIOTECHNOLOGY CORPORATION (US) 1998-04-02 WO disclosed