SCHEMBL8445858

SCHEMBL8445858

Cc1cn(CCCN2C(=O)c3ccccc3C2=O)c(Cc2ccccc2)n1

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
MAOB P27338 5/20 0.46
ACHE P22303 10/20 0.44
BCHE P06276 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6494289 0.81 RXFP1 (0.55)
SCHEMBL8443893 0.79 TLR8 (0.44)
SCHEMBL4351612 0.71 TDP1 (0.66) TDP1L3MBTL1
SCHEMBL28062278 0.70 RXFP1 (0.42) TDP1
SCHEMBL45050 0.68 TDP1 (0.86) TDP1L3MBTL1MAOBACHE
SCHEMBL30371663 0.68 TDP1 (0.86) TDP1L3MBTL1MAOBACHE
SCHEMBL8445961 0.68 CREBBP (0.50)
SCHEMBL3040144 0.68 ALDH1A1 (0.53)
SCHEMBL661168 0.68 QPCT (0.52)
SCHEMBL661173 0.68 QPCT (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618907-B1 1-(ARYLALKYL-AMINOALKYL)IMIDAZOLE DERIVATIVES, PROCESSES OF PREPARATION AND USE AS THERAPEUTICAL AGENTS BRITISH TECH GROUP INT (GB) 1999-04-28 EP disclosed
US-5547972-A 1-(ARLALKYLAMINOALKYL) IMIDAZOLE DERIVATIVES THE BOOTS COMPANY PLC (GB) 1996-08-20 US disclosed
EP-0618907-A1 1-(ARYLALKYL-AMINOALKYL)IMIDAZOLE DERIVATIVES, PROCESSES OF PREPARATION AND USE AS THERAPEUTICAL AGENTS Knoll AG (DE) 1994-10-12 EP disclosed
WO-1993013075-A1 1-(ARYLALKYL-AMINOALKYL)IMIDAZOLE DERIVATIVES, PROCESSES OF PREPARATION AND USE AS THERAPEUTICAL AGENTS THE BOOTS COMPANY PLC (GB) 1993-07-08 WO disclosed