SCHEMBL8447293

SCHEMBL8447293

CC1(C)c2cc(Br)cc(Br)c2Oc2c(Br)cc(Br)cc21

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AHR P35869 2/20 0.50
ALOX15 P16050 2/20 0.38
ALOX12 P18054 2/20 0.38
CYP3A4 P08684 1/20 0.32
TSHR P16473 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
MEN1 O00255 1/20 0.31
CRHBP P24387 1/20 0.31
KMT2A Q03164 1/20 0.31
CRHR2 Q13324 1/20 0.31
DRD1 P21728 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL708899 0.76 GABBR2 (0.36) AHRALOX15ALOX12CYP3A4TSHR
SCHEMBL2489432 0.71 AHR (0.38) AHRALOX15ALOX12
SCHEMBL30153513 0.70 DRD1 (0.49) DRD1
SCHEMBL16146962 0.70 DRD1 (0.49) DRD1
SCHEMBL8163979 0.69 PRMT1 (0.50) ALOX15ALOX12CYP3A4TSHRTDP1
SCHEMBL2856011 0.65
SCHEMBL15841475 0.65 AHR (0.54) AHR
SCHEMBL30153529 0.65 AHR (0.54) AHR
SCHEMBL3685579 0.65 AHR (0.33) AHR
SCHEMBL12440926 0.64 PGR (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5877030-A REACTING AMINO ACID MOLECULES WITH REACTIVE XANTHENE DERIVATIVES, COMBINATORIAL LIBRARIES SILICON VALLEY BANK 1999-03-02 US disclosed
WO-1995019359-A1 PROCESS FOR MAKING XANTHENE OR CUBANE BASED COMPOUNDS, AND PROTEASE INHIBITORS MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 1995-07-20 WO disclosed