SCHEMBL8450784

SCHEMBL8450784

CON(C)C(=O)C1CCc2cc3ccccc3n2C1

nearest known ligand 0.39

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.39
HTR2C P28335 4/20 0.39
SIGMAR1 Q99720 7/20 0.37
MCL1 Q07820 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8446842 0.89 HTR2A (0.44) HTR2AHTR2CSIGMAR1
SCHEMBL8453122 0.88 SIGMAR1 (0.38) HTR2AHTR2CSIGMAR1MCL1
SCHEMBL21027979 0.83 HTR2A (0.43) HTR2AHTR2CSIGMAR1
SCHEMBL8448530 0.81 SIGMAR1 (0.42) HTR2AHTR2CSIGMAR1
SCHEMBL8447696 0.79 HTR2A (0.43) HTR2AHTR2CSIGMAR1
SCHEMBL8450915 0.78 HTR2A (0.43) HTR2AHTR2CSIGMAR1
SCHEMBL8328343 0.77 ALDH1A1 (0.45) HTR2AHTR2C
SCHEMBL8658423 0.73 HTR2A (0.43) HTR2AHTR2CSIGMAR1
SCHEMBL8656153 0.71 HTR2A (0.41) HTR2AHTR2CSIGMAR1
SCHEMBL233436 0.70 HTR2A (0.47) HTR2AHTR2CSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0624586-B1 Substituted pyrroles HOFFMANN LA ROCHE (CH) 1999-09-01 EP disclosed
US-5721230-A ANTIINFLAMMATORY AGENT, VIRICIDES; TREATING CARDIOVASCULAR DISORDER, RESPIRATORY SYSTEM DISORDER, THROMBOSIS, DIABETES, ALOPECIA HOFFMANN-LA ROCHE INC. (US) 1998-02-24 US disclosed
EP-0624586-A1 Substituted pyrroles F. HOFFMANN-LA ROCHE AG (CH) 1994-11-17 EP disclosed