SCHEMBL844919

SCHEMBL844919

CC(C)(C)C(=O)N1CCC[C@H]1C(=O)Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3CCCN3C(=O)C(C)(C)C)cc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.54
EP300 Q09472 2/20 0.53
CREBBP Q92793 2/20 0.53
HTT P42858 2/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
ALDH1A1 P00352 3/20 0.47
MAPK1 P28482 2/20 0.47
RHOC P08134 1/20 0.46
RHOA P61586 1/20 0.46
PABPC1 P11940 1/20 0.45
TSHR P16473 1/20 0.45
LMNA P02545 1/20 0.44
RIPK1 Q13546 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL844899 0.85 NPC1 (0.52) NPC1EP300CREBBPHTTCYP2C9
SCHEMBL845452 0.85 F2 (0.52) NPC1EP300CREBBPHTTCYP2C9
SCHEMBL10299164 0.84 NPC1 (0.76) NPC1EP300CREBBPHTTCYP2C9
SCHEMBL10281278 0.84 NPC1 (0.76) NPC1EP300CREBBPHTTCYP2C9
SCHEMBL845227 0.84 NPC1 (0.76) NPC1EP300CREBBPHTTCYP2C9
SCHEMBL845258 0.84 MAPK1 (0.60) NPC1EP300CREBBPHTTCYP2C9
SCHEMBL845774 0.82 CYP2C19 (0.49) NPC1EP300CREBBPHTTCYP2C9
SCHEMBL845251 0.82 PABPC1 (0.50) NPC1EP300CREBBPHTTCYP2C9
SCHEMBL844894 0.82 CYP2C19 (0.55) NPC1HTTCYP2C9CYP2C19MEN1
SCHEMBL844890 0.82 KCNH2 (0.51) NPC1HTTCYP2C9CYP2C19MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed