SCHEMBL845000

SCHEMBL845000

COc1ccc(Cl)cc1C(=O)N1CCC[C@H]1C(=O)Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3CCCN3C(=O)c3cc(Cl)ccc3OC)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RHOC P08134 1/20 0.51
RHOA P61586 1/20 0.51
EP300 Q09472 6/20 0.51
CREBBP Q92793 6/20 0.51
TSHR P16473 1/20 0.50
SMN1; SMN2 Q16637 2/20 0.48
MAPK1 P28482 1/20 0.48
ALDH1A1 P00352 2/20 0.48
MAPT P10636 1/20 0.48
ROCK2 O75116 1/20 0.47
LMNA P02545 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845629 0.97 TSHR (0.50) RHOCRHOAEP300CREBBPTSHR
SCHEMBL845290 0.91 HCRTR1 (0.52) TSHRSMN1; SMN2MAPK1ALDH1A1MAPT
SCHEMBL845002 0.89 CYP2C9 (0.55) EP300CREBBPTSHRSMN1; SMN2MAPK1
SCHEMBL845539 0.87 HCRTR1 (0.54) EP300CREBBPTSHRSMN1; SMN2MAPK1
SCHEMBL845284 0.86 MAPK1 (0.58) EP300CREBBPMAPK1ALDH1A1ROCK2
SCHEMBL873856 0.83 HCRTR1 (0.45) TSHRSMN1; SMN2MAPK1ALDH1A1MAPT
SCHEMBL873577 0.82 LMNA (0.47) EP300CREBBPTSHRSMN1; SMN2MAPK1
SCHEMBL13272181 0.82 MAPK1 (0.53) EP300CREBBPMAPK1ALDH1A1ROCK2
SCHEMBL845641 0.82 MAPK1 (0.53) EP300CREBBPMAPK1ALDH1A1ROCK2
SCHEMBL874313 0.78 MAPK1 (0.50) EP300CREBBPTSHRMAPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed