SCHEMBL873577

SCHEMBL873577

COc1ccc(OC)c(C(=O)N2CCC[C@H]2C(=O)Nc2ccc(/C=C/c3ccc(NC(=O)[C@@H]4CCCN4)cc3)cc2)c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.47
HPGD P15428 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
TSHR P16473 1/20 0.46
MAPK1 P28482 2/20 0.46
ALDH1A1 P00352 2/20 0.46
HTT P42858 1/20 0.46
GFER P55789 1/20 0.44
HCRTR1 O43613 1/20 0.44
HCRTR2 O43614 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
EP300 Q09472 3/20 0.43
CREBBP Q92793 3/20 0.43
TDP1 Q9NUW8 1/20 0.43
TP53 P04637 1/20 0.42
ROCK2 O75116 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL873856 0.93 HCRTR1 (0.45) SMN1; SMN2CYP2C9CYP2C19TSHRMAPK1
SCHEMBL845002 0.91 CYP2C9 (0.55) LMNAHPGDSMN1; SMN2CYP2C9CYP2C19
SCHEMBL874313 0.89 MAPK1 (0.50) LMNACYP2C9CYP2C19TSHRMAPK1
SCHEMBL845539 0.89 HCRTR1 (0.54) LMNAHPGDSMN1; SMN2CYP2C9CYP2C19
SCHEMBL10119619 0.85 MAPK1 (0.46) LMNACYP2C9CYP2C19MAPK1ALDH1A1
SCHEMBL845290 0.84 HCRTR1 (0.52) LMNAHPGDSMN1; SMN2CYP2C9CYP2C19
SCHEMBL873862 0.82 ALDH1A1 (0.45) LMNACYP2C9CYP2C19TSHRMAPK1
SCHEMBL845000 0.82 RHOC (0.51) LMNASMN1; SMN2CYP2C9CYP2C19TSHR
SCHEMBL872930 0.80 GAA (0.52) LMNACYP2C9CYP2C19TSHRMAPK1
SCHEMBL874324 0.80 MAPK1 (0.42) LMNACYP2C9CYP2C19MAPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed