SCHEMBL8451632

SCHEMBL8451632

C#Cc1cccc(Nc2ncnc3cnc(N(C)C4CCN(C)CC4)nc23)c1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BRAF P15056 5/20 0.52
EGFR P00533 14/20 0.51
ERBB2 P04626 2/20 0.47
ERBB4 Q15303 1/20 0.47
HPGD P15428 1/20 0.46
HTT P42858 1/20 0.46
FBP1 P09467 2/20 0.43
GAK O14976 2/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
RIPK2 O43353 1/20 0.41
BUB1 O43683 1/20 0.41
STK10 O94804 1/20 0.41
CARS1 P49589 1/20 0.41
MAP3K1 Q13233 1/20 0.41
PIP4K2C Q8TBX8 1/20 0.41
SLK Q9H2G2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6993268 0.91 BRAF (0.55) BRAFEGFRERBB2HPGDHTT
SCHEMBL8318037 0.89 EGFR (0.52) BRAFEGFRERBB2ERBB4FBP1
SCHEMBL6997891 0.85 BRAF (0.56) BRAFEGFRERBB2HPGDHTT
SCHEMBL8316279 0.84 EGFR (0.65) BRAFEGFRERBB2ERBB4HPGD
SCHEMBL7578315 0.84 BRAF (0.45) BRAFEGFRERBB2ERBB4FBP1
SCHEMBL6996263 0.83 BRAF (0.51) BRAFEGFRERBB2HPGDHTT
SCHEMBL6997218 0.82 BRAF (0.50) BRAFEGFRERBB2HPGDHTT
SCHEMBL6996275 0.82 EGFR (0.60) BRAFEGFRERBB2HPGDHTT
SCHEMBL6986988 0.80 EGFR (0.72) BRAFEGFRERBB2ERBB4HPGD
SCHEMBL8319176 0.78 CSNK2A1 (0.53) BRAFEGFRERBB2HPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888351-A1 PYRIMIDO 5,4-D]PYRIMIDINES, MEDICAMENTS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESS FOR THEIR PRODUCTION Dr. Karl Thomae GmbH (DE) 1999-01-07 EP disclosed
WO-1997032880-A1 PYRIMIDO[5,4-D]PYRIMIDINES, MEDICAMENTS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESS FOR THEIR PRODUCTION DR. KARL THOMAE GMBH (DE) 1997-09-12 WO disclosed