SCHEMBL8452234

SCHEMBL8452234

O=C(N(CCOc1cccc([AsH2])c1[AsH2])Cc1cccc2ccccc12)C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.41
ALDH1A1 P00352 3/20 0.41
HTR1B P28222 7/20 0.38
HPGD P15428 2/20 0.38
ATM Q13315 1/20 0.38
TSHR P16473 1/20 0.37
HTR1D P28221 3/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
CDYL Q9Y232 1/20 0.36
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
SLC6A9 P48067 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7333407 0.83 KDM4E (0.41) KDM4EALDH1A1HTR1BHPGDATM
SCHEMBL7343282 0.81 KCNH2 (0.39) KDM4EALDH1A1HPGDATMMEN1
SCHEMBL7337149 0.79 DRD2 (0.44) KDM4EALDH1A1HTR1BHPGDATM
SCHEMBL8344355 0.79 DRD2 (0.43) KDM4EALDH1A1HTR1BHPGDATM
SCHEMBL17513639 0.71 METAP2 (0.44) HDAC1HDAC6NPSR1
SCHEMBL16899094 0.69 METAP2 (0.44) HDAC1HDAC6
SCHEMBL16899167 0.67 METAP2 (0.45) HDAC1HDAC6
SCHEMBL7334771 0.66 KDM4E (0.42) KDM4EALDH1A1HTR1BHTR1DL3MBTL1
SCHEMBL16899264 0.65 MC4R (0.42) KMT2AHDAC1HDAC6
SCHEMBL11374514 0.65 KDM4E (0.47) KDM4EALDH1A1HTR1BHPGDATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0964854-A1 4-AMINOALKOXY-1,3-DIHYDROBENZOIMIDAZOL-2-THIONES DERIVATIVES, THEIR PREPARATION AND THEIR USE AS DOPAMINE AUTORECEPTOR (D2) AGONISTS AMERICAN HOME PRODUCTS CORPORATION (US) 1999-12-22 EP disclosed
WO-1998035947-A1 4-AMINOALKOXY-1,3-DIHYDROBENZOIMIDAZOL-2-THIONES DERIVATIVES, THEIR PREPARATION AND THEIR USE AS DOPAMINE AUTORECEPTOR (D2) AGONISTS AMERICAN HOME PRODUCTS CORPORATION (US) 1998-08-20 WO disclosed