SCHEMBL845453

SCHEMBL845453

O=C(Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3CCCN3C(=O)N3CCOCC3)cc2)cc1)[C@@H]1CCCN1C(=O)N1CCOCC1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 4/20 0.53
ALDH1A1 P00352 4/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
HTT P42858 2/20 0.44
NPC1 O15118 1/20 0.43
MAPK1 P28482 1/20 0.43
EP300 Q09472 1/20 0.42
CREBBP Q92793 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
RHOC P08134 1/20 0.41
RHOA P61586 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845170 0.90 CYP2C9 (0.47) CNR2ALDH1A1CYP2C9CYP2C19HTT
SCHEMBL844884 0.79 HTT (0.48) ALDH1A1CYP2C9CYP2C19HTTNPC1
SCHEMBL28434981 0.78 CNR2 (0.46) CNR2ALDH1A1CYP2C9CYP2C19HTT
SCHEMBL28434982 0.78 CNR2 (0.46) CNR2ALDH1A1CYP2C9CYP2C19HTT
SCHEMBL845500 0.78 HPGD (0.51) ALDH1A1CYP2C9NPC1MEN1KMT2A
SCHEMBL845495 0.78 HPGD (0.51) ALDH1A1CYP2C9NPC1MEN1KMT2A
SCHEMBL845258 0.78 MAPK1 (0.60) ALDH1A1CYP2C9CYP2C19HTTNPC1
SCHEMBL845255 0.78 CYP2C9 (0.47) CNR2ALDH1A1CYP2C9CYP2C19HTT
SCHEMBL845774 0.77 CYP2C19 (0.49) ALDH1A1CYP2C9CYP2C19HTTNPC1
SCHEMBL873200 0.77 RHOC (0.48) ALDH1A1CYP2C9CYP2C19HTTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed