SCHEMBL8457641

SCHEMBL8457641

O=c1cc2oc3ccccc3cc-2c([N+](=O)[O-])c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.51
LMNA P02545 2/20 0.51
MAOB P27338 5/20 0.44
RAB9A P51151 3/20 0.43
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
GABRP O00591 1/20 0.43
GABRD O14764 1/20 0.43
GABRA1 P14867 1/20 0.43
GABRB1 P18505 1/20 0.43
GABRG2 P18507 1/20 0.43
GABRB3 P28472 1/20 0.43
GABRA5 P31644 1/20 0.43
GABRA3 P34903 1/20 0.43
GABRA2 P47869 1/20 0.43
GABRB2 P47870 1/20 0.43
GABRA4 P48169 1/20 0.43
GABRE P78334 1/20 0.43
GABRA6 Q16445 1/20 0.43
GABRG1 Q8N1C3 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6156827 0.86 ALDH1A1 (0.56) ALDH1A1LMNAMAOBRAB9AKMT2A
SCHEMBL27687599 0.82 TNKS (0.52) ALDH1A1MAOBRAB9AKMT2AMEN1
SCHEMBL9754513 0.80 ALDH1A1 (0.67) ALDH1A1LMNAMAOBRAB9AKMT2A
SCHEMBL6896489 0.79 ALDH1A1 (0.48) ALDH1A1LMNAMAOBRAB9AKMT2A
SCHEMBL28506238 0.78 ALDH1A1 (0.52) ALDH1A1LMNAMAOBRAB9AKMT2A
SCHEMBL5941127 0.76 HPGD (0.56) ALDH1A1LMNAMAOBRAB9AKMT2A
SCHEMBL30422441 0.76 HPGD (0.56) ALDH1A1LMNAMAOBRAB9AKMT2A
SCHEMBL9238022 0.76 RAB9A (0.49) ALDH1A1LMNAMAOBRAB9AKMT2A
SCHEMBL8868150 0.75 KMT2A (0.48) ALDH1A1LMNAMAOBRAB9AKMT2A
SCHEMBL8583022 0.75 RAB9A (0.48) ALDH1A1LMNAMAOBRAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934270-A1 A METHOD OF TREATING CANCER Merck & Co., Inc. (US) 1999-08-11 EP disclosed
WO-1997045412-A1 A METHOD OF TREATING CANCER MERCK & CO., INC. (US) 1997-12-04 WO disclosed