SCHEMBL8458765

SCHEMBL8458765

COc1ccccc1C[C@H](C[C@H](O[Si](C)(C)C(C)(C)C)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 1/20 0.48
ITGB7 P26010 1/20 0.48
KLK5 Q9Y337 3/20 0.43
ALDH1A1 P00352 4/20 0.41
GAA P10253 1/20 0.41
TACR1 P25103 1/20 0.40
ATM Q13315 1/20 0.40
PSEN1 P49768 3/20 0.40
PSEN2 P49810 3/20 0.40
APH1B Q8WW43 3/20 0.40
NCSTN Q92542 3/20 0.40
APH1A Q96BI3 3/20 0.40
PSENEN Q9NZ42 3/20 0.40
ACE P12821 1/20 0.39
APP P05067 1/20 0.39
CTSS P25774 2/20 0.39
CTSL P07711 1/20 0.39
CTSB P07858 1/20 0.39
CTSK P43235 1/20 0.39
LMNA P02545 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8853318 1.00 ITGA4 (0.48) ITGA4ITGB7KLK5ALDH1A1GAA
SCHEMBL7627308 0.91 KLK5 (0.42) ITGA4ITGB7KLK5ALDH1A1ATM
SCHEMBL7627313 0.91 KLK5 (0.42) ITGA4ITGB7KLK5ALDH1A1ATM
SCHEMBL7629868 0.90 KLK5 (0.41) ITGA4ITGB7KLK5ALDH1A1ATM
SCHEMBL7633741 0.90 KLK5 (0.41) ITGA4ITGB7KLK5ALDH1A1ATM
SCHEMBL7629875 0.90 KLK5 (0.41) ITGA4ITGB7KLK5ALDH1A1ATM
SCHEMBL7633738 0.90 KLK5 (0.41) ITGA4ITGB7KLK5ALDH1A1ATM
SCHEMBL6305846 0.90 KLK5 (0.47) KLK5ALDH1A1ATMPSEN1PSEN2
SCHEMBL7283432 0.90 KLK5 (0.47) KLK5ALDH1A1ATMPSEN1PSEN2
SCHEMBL6446803 0.90 KLK5 (0.47) KLK5ALDH1A1ATMPSEN1PSEN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5935976-A Antiviral ethers of aspartate protease substrate isosteres NOVARTIS CORPORATION (US) 1999-08-10 US disclosed
US-5807891-A RETROVIRUSES NOVARTIS AG (CH) 1998-09-15 US disclosed
US-5663200-A CARBAMOYL PEPTIDE DERIVATIVES AS VIRICIDES CIBA-GEIGY CORPORATION (US) 1997-09-02 US disclosed
US-5643878-A TREATMENT OF RETROVIRAL DISEASES LIKE AIDS CIBA-GEIGY CORPORATION (US) 1997-07-01 US disclosed
EP-0708085-A2 Antiviral ethers of aspartate protease substrate isosteres CIBA-GEIGY AG (CH) 1996-04-24 EP disclosed