SCHEMBL8459092

SCHEMBL8459092

CC(C)(C)OC(=O)C(CNC(=O)c1ccccc1)NS(=O)(=O)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 8/20 0.56
ITGB3 P05106 12/20 0.55
ITGA2B P08514 11/20 0.55
PSMB8 P28062 1/20 0.48
PSMB5 P28074 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7490103 0.93 ITGB3 (0.53) ITGAVITGB3ITGA2B
SCHEMBL8903718 0.93 ITGB3 (0.53) ITGAVITGB3ITGA2B
SCHEMBL8902514 0.90 ITGAV (0.52) ITGAVITGB3ITGA2BPSMB8PSMB5
SCHEMBL7486439 0.85 ITGB3 (0.60) ITGAVITGB3ITGA2B
SCHEMBL7377406 0.85 ITGB3 (0.48) ITGAVITGB3ITGA2BPSMB8
SCHEMBL6493323 0.85 ITGB3 (0.48) ITGAVITGB3ITGA2B
SCHEMBL6492757 0.85 ITGB3 (0.48) ITGAVITGB3ITGA2B
SCHEMBL7493829 0.84 ITGB3 (0.61) ITGAVITGB3ITGA2B
SCHEMBL7495217 0.84 ITGB3 (0.54) ITGAVITGB3ITGA2B
SCHEMBL383058 0.83 ITGB3 (0.58) ITGAVITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5929120-A Guainidino, formamidino, amino and related compounds for inhibiting osteoclast-mediated bone resorption MERCK & CO., INC. (US) 1999-07-27 US disclosed
US-5741796-A Pyridyl and naphthyridyl compounds for inhibiting osteoclast-mediated bone resorption MERCK & CO., INC. (US) 1998-04-21 US disclosed