SCHEMBL8465223

SCHEMBL8465223

Oc1ccc2c(c1)[C@H](O)[C@@H](Oc1ccccc1)CC2

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.41
ESR2 Q92731 1/20 0.41
DRD1 P21728 5/20 0.41
DRD2 P14416 2/20 0.41
HTR2A P28223 1/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2B Q13224 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8465230 1.00 ESR1 (0.41) ESR1ESR2DRD1DRD2HTR2A
SCHEMBL8465226 1.00 ESR1 (0.41) ESR1ESR2DRD1DRD2HTR2A
SCHEMBL8465149 0.83 KDM1A (0.50) HTR2A
SCHEMBL8465154 0.83 KDM1A (0.50) HTR2A
SCHEMBL8464032 0.77 DRD3 (0.38) ESR1ESR2DRD2GRIN1GRIN2B
SCHEMBL8464035 0.77 DRD3 (0.38) ESR1ESR2DRD2GRIN1GRIN2B
SCHEMBL8464040 0.77 DRD3 (0.38) ESR1ESR2DRD2GRIN1GRIN2B
SCHEMBL8466002 0.74 CYSLTR1 (0.54)
SCHEMBL8348051 0.74 ALOX5 (0.38)
SCHEMBL8348060 0.74 ALOX5 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5998451-A LIPOXYGENASE INHIBITORS PFIZER INC (US) 1999-12-07 US disclosed
US-5059609-A Lipoxygenase inhibitors; leukotriene receptor blockers; psoriasis; antiulcer agents and myocardial infarctions PFIZER INC. (US) 1991-10-22 US disclosed
EP-0313295-A2 Substituted tetralins, chromans and related compounds in the treatment of asthma, arthritis and related diseases PFIZER INC. (US) 1989-04-26 EP disclosed