SCHEMBL8466376

SCHEMBL8466376

CC(C)(CO)CO.COc1ccc(C=C(C(=O)O)C(=O)O)cc1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.45
ATM Q13315 1/20 0.45
GSK3B P49841 2/20 0.44
PPARA Q07869 1/20 0.44
AKR1C3 P42330 1/20 0.44
MAPT P10636 3/20 0.44
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 2/20 0.44
HPGD P15428 2/20 0.44
TP53 P04637 1/20 0.44
F3 P13726 1/20 0.42
RAB9A P51151 2/20 0.42
NPC1 O15118 1/20 0.42
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 1/20 0.41
TSHR P16473 1/20 0.41
NFKB1 P19838 1/20 0.41
APEX1 P27695 1/20 0.41
BLM P54132 1/20 0.41
PMP22 Q01453 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL433921 0.87 THRB (0.56) THRBATMGSK3BAKR1C3MAPT
Hydrochloric Acid SCHEMBL8581964 0.85 THRB (0.55) THRBATMGSK3BAKR1C3MAPT
SCHEMBL7820837 0.84 THRB (0.56) THRBATMGSK3BAKR1C3MAPT
SCHEMBL7820839 0.84 THRB (0.56) THRBATMGSK3BAKR1C3MAPT
SCHEMBL9476783 0.79 ALDH1A1 (0.53) THRBATMGSK3BAKR1C3MAPT
SCHEMBL9476792 0.79 ALDH1A1 (0.53) THRBATMGSK3BAKR1C3MAPT
SCHEMBL16166799 0.78 KMT2A (0.44) THRBATMGSK3BPPARAAKR1C3
SCHEMBL5645074 0.78 THRB (0.50) THRBATMGSK3BAKR1C3MAPT
SCHEMBL1514195 0.78 THRB (0.50) THRBATMGSK3BAKR1C3MAPT
SCHEMBL6380249 0.76 THRB (0.49) THRBATMGSK3BAKR1C3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5916942-A COATING WHICH PROTECTS AGAINST THE EFFECT OF ULTRAVIOLET RADIATION AND PREVENTS THE FORMATION OF WATER DROPLETS BAYER AG (DE) 1999-06-29 US disclosed
US-4588807-A ANTIASTHMA, ANTIULCERE, ANTICOAGULANT BAYER AKTIENGESELLSCHAFT (DE) 1986-05-13 US disclosed