SCHEMBL8466508

SCHEMBL8466508

CCCCCc1[nH]nc2ncnc(Cl)c12

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RPS6KB1 P23443 12/20 0.42
PI4KA P42356 1/20 0.38
PI4K2B Q8TCG2 1/20 0.38
PI4K2A Q9BTU6 1/20 0.38
PI4KB Q9UBF8 1/20 0.38
PAK1 Q13153 1/20 0.35
PBRM1 Q86U86 1/20 0.35
HTT P42858 1/20 0.33
NCOA1 Q15788 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NCOA3 Q9Y6Q9 1/20 0.33
ABL1 P00519 1/20 0.33
SRC P12931 1/20 0.33
AKT1 P31749 2/20 0.32
AKT2 P31751 1/20 0.32
RPS6KA3 P51812 1/20 0.32
HCAR2 Q8TDS4 3/20 0.31
HCAR3 P49019 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8466427 0.82 PI4KB (0.50) PI4KAPI4K2BPI4K2API4KBABL1
SCHEMBL8466511 0.74 CHEK1 (0.36) PI4KAPI4K2BPI4K2API4KBPAK1
SCHEMBL6273819 0.71 PI4KA (0.35) PI4KAPI4K2BPI4K2API4KBPAK1
SCHEMBL6431494 0.70 RPS6KB1 (0.46) RPS6KB1ABL1SRCAKT1AKT2
SCHEMBL3322337 0.69 TYMP (0.39) PI4KAPI4K2BPI4K2API4KBPAK1
SCHEMBL4453790 0.68 TYMP (0.41) PI4KAPI4K2BPI4K2API4KBSMN1; SMN2
SCHEMBL1129156 0.67 AURKA (0.38) RPS6KB1SRC
SCHEMBL900339 0.64 MAPT (0.43) HTTSMN1; SMN2RPS6KA3
SCHEMBL12495916 0.63 ALDH1A1 (0.39) HTTSMN1; SMN2
SCHEMBL1128852 0.62 CHEK1 (0.40) ABL1SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0496617-B1 Adenosine kinase inhibitors METABASIS THERAPEUTICS INC (US) 1999-12-01 EP disclosed
US-5646128-A TREATING INFLAMMATION, SEPSIS, SEPTIC SHOCK, BURNS GENSIA, INC. (US) 1997-07-08 US disclosed
WO-1994017803-A9 ADENOSINE KINASE INHIBITORS 1994-09-29 WO disclosed
WO-1992012718-A1 ADENOSINE KINASE INHIBITORS GENSIA, INC. (US) 1992-08-06 WO disclosed
EP-0496617-A1 Adenosine kinase inhibitors GENSIA, INC. (US) 1992-07-29 EP disclosed