L-768673

L-768673

SCHEMBL8466533

CCOP(=O)(OCC)SCCSCC.O=C(Cc1ccc(C(F)(F)F)cc1C(F)(F)F)N[C@@H]1N=C(c2ccccc2)c2ccccc2N(CC(F)(F)F)C1=O

nearest known ligand 0.74

Full drug profile on Sugi Atlas →

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.74
CALCRL Q16602 14/20 0.47
CCKAR P32238 2/20 0.43
CCKBR P32239 2/20 0.43
RAMP1 O60894 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
L-768673 SCHEMBL7207125 0.86 KCNH2 (1.00) KCNH2CALCRLCCKARCCKBRRAMP1
SCHEMBL7965787 0.82 KCNH2 (0.85) KCNH2CALCRLCCKARCCKBRRAMP1
SCHEMBL8745076 0.81 KCNH2 (0.89) KCNH2CALCRLRAMP1
SCHEMBL7744138 0.79 KCNH2 (0.80) KCNH2CALCRLCCKARCCKBR
SCHEMBL8462992 0.78 KCNH2 (0.82) KCNH2CALCRLRAMP1
SCHEMBL8820683 0.76 KCNH2 (0.77) KCNH2CCKARCCKBR
SCHEMBL8760273 0.75 KCNH2 (0.75) KCNH2CALCRLCCKARCCKBRRAMP1
SCHEMBL7744135 0.75 KCNH2 (0.72) KCNH2CCKARCCKBR
SCHEMBL7744593 0.75 KCNH2 (0.72) KCNH2CCKARCCKBR
SCHEMBL8462904 0.75 KCNH2 (0.77) KCNH2CALCRLCCKARCCKBRRAMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0776208-B1 2,3-DIHYDRO-1-(2,2,2-TRIFLUOROETHYL)-2-OXO-5-PHENYL-1H-1,4-BENZODIAZEPINES MERCK & CO INC (US) 1999-11-10 EP claimed