SCHEMBL8467175

SCHEMBL8467175

CC(C)c1cc(-c2ccc(F)c3ccccc23)nc(S(C)(=O)=O)n1.[H+]

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1B P28222 1/20 0.63
HTR2B P41595 1/20 0.63
GPR65 Q8IYL9 1/20 0.63
LMNA P02545 5/20 0.42
KDM4E B2RXH2 5/20 0.42
KMT2A Q03164 4/20 0.42
ALDH1A1 P00352 4/20 0.42
SDHB P21912 7/20 0.41
BPTF Q12830 2/20 0.39
NPSR1 Q6W5P4 5/20 0.39
STAT3 P40763 4/20 0.39
HPGD P15428 4/20 0.39
HTT P42858 4/20 0.39
MITF O75030 2/20 0.39
RAB9A P51151 4/20 0.38
TP53 P04637 3/20 0.38
HSD17B10 Q99714 3/20 0.38
STAT1 P42224 2/20 0.38
TLR9 Q9NR96 2/20 0.38
S1PR4 O95977 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5748949 0.99 HTR1B (0.64) HTR1BHTR2BGPR65LMNAKDM4E
SCHEMBL5745041 0.82 HTR1B (0.45) HTR1BHTR2BGPR65LMNAKDM4E
SCHEMBL5746388 0.81 HTR1B (0.64) HTR1BHTR2BGPR65KDM4ENPSR1
SCHEMBL5749062 0.81 HTR1B (0.60) HTR1BHTR2BGPR65ALOX5APFEN1
SCHEMBL8469545 0.79 HTR1B (0.97) HTR1BHTR2BGPR65ALOX5APFEN1
SCHEMBL18461518 0.79 HTR1B (0.72) HTR1BHTR2BGPR65ALOX5APFEN1
SCHEMBL5749278 0.79 LMNA (0.53) HTR1BHTR2BGPR65LMNAKDM4E
SCHEMBL375979 0.78 HTR1B (1.00) HTR1BHTR2BGPR65ALOX5APFEN1
SCHEMBL8382821 0.78 HTR1B (0.71) HTR1BHTR2BGPR65ALOX5APFEN1
SCHEMBL5751060 0.77 HTR1B (0.41) HTR1BHTR2BGPR65LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0901474-A1 ARYL PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-03-17 EP disclosed
WO-1997044326-A1 ARYL PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-11-27 WO disclosed