SCHEMBL8467358

SCHEMBL8467358

CC(C)=CCc1cc(/C=C/C(=O)O)cc(O)c1O

nearest known ligand 0.86

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 10/20 0.86
AKR1B10 O60218 2/20 0.86
AKR1B1 P15121 2/20 0.86
MMP2 P08253 1/20 0.86
PAK1 Q13153 1/20 0.86
ALOX5 P09917 2/20 0.58
PTGES O14684 1/20 0.58
NFKB1 P19838 1/20 0.58
STAT3 P40763 1/20 0.58
NFKB2 Q00653 1/20 0.58
RELA Q04206 1/20 0.58
PTPN1 P18031 5/20 0.57
AKR1C2 P52895 8/20 0.56
OSBP P22059 1/20 0.55
MGAM O43451 1/20 0.48
MAOA P21397 1/20 0.48
MAOB P27338 1/20 0.48
XDH P47989 1/20 0.48
AKR1C4 P17516 1/20 0.47
PTGS1 P23219 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8467360 1.00 AKR1C3 (0.86) AKR1C3AKR1B10AKR1B1MMP2PAK1
Artepillin SCHEMBL2138507 0.92 AKR1C3 (1.00) AKR1C3AKR1B10AKR1B1MMP2PAK1
Artepillin SCHEMBL7128580 0.92 AKR1C3 (1.00) AKR1C3AKR1B10AKR1B1MMP2PAK1
Artepillin SCHEMBL1229229 0.92 AKR1C3 (1.00) AKR1C3AKR1B10AKR1B1MMP2PAK1
SCHEMBL25890163 0.88 AKR1C3 (0.91) AKR1C3AKR1B10AKR1B1MMP2PAK1
SCHEMBL26422962 0.88 AKR1C3 (0.91) AKR1C3AKR1B10AKR1B1MMP2PAK1
SCHEMBL23742688 0.85 AKR1C3 (0.84) AKR1C3AKR1B10AKR1B1MMP2PAK1
SCHEMBL11036838 0.85 AKR1C3 (0.84) AKR1C3AKR1B10AKR1B1MMP2PAK1
SCHEMBL29574915 0.85 AKR1C3 (0.84) AKR1C3AKR1B10AKR1B1MMP2PAK1
SCHEMBL23742687 0.85 AKR1C3 (0.84) AKR1C3AKR1B10AKR1B1MMP2PAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114377006-B Absorption promoter for cinnamic acid derivative 株式会社山田养蜂场本社 2024-02-09 CN claimed
CN-114377006-A Absorption enhancer for cinnamic acid derivatives 株式会社山田养蜂场本社 2022-04-22 CN claimed
US-20220105054-A1 ABSORPTION ENHANCER OF CINNAMIC ACID DERIVATIVE YAMADA BEE COMPANY, INC. (JP) 2022-04-07 US claimed
JP-11349526-A None JP disclosed
CN-114377006-B Absorption promoter for cinnamic acid derivative 株式会社山田养蜂场本社 2024-02-09 CN disclosed
CN-114377006-A Absorption enhancer for cinnamic acid derivatives 株式会社山田养蜂场本社 2022-04-22 CN disclosed
US-20220105054-A1 ABSORPTION ENHANCER OF CINNAMIC ACID DERIVATIVE YAMADA BEE COMPANY, INC. (JP) 2022-04-07 US disclosed
JP-H11349526-A NEW COMPOUND OR ITS PHARMACOLOGICALLY ACCEPTABLE SALT AND ANTIOXIDANT CONTAINING THE SAME AS ACTIVE INGREDIENT OYO SEIKAGAKU KENKYUSHO 1999-12-21 JP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220105054-A1 ABSORPTION ENHANCER OF CINNAMIC ACID DERIVATIVE FABP2, SLC16A3, SLC16A7 AKR1C3 261/4885AKR1B10 583/4885AKR1B1 363/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.