SCHEMBL8467480

SCHEMBL8467480

C[Si](C)(NC(=O)c1ccccc1)C1=CC=CC1.[LiH].[LiH]

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
IDO1 P14902 1/20 0.38
ALOX15 P16050 1/20 0.38
HDAC1 Q13547 1/20 0.38
CA9 Q16790 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HSD17B10 Q99714 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
NCOR2 Q9Y618 1/20 0.38
NPC1 O15118 5/20 0.37
RAB9A P51151 5/20 0.37
KMT2A Q03164 4/20 0.37
ALDH1A1 P00352 4/20 0.37
MEN1 O00255 3/20 0.37
MAPT P10636 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7633339 0.74 NPC1 (0.38) HDAC3CA12CA1IDO1ALOX15
SCHEMBL8467168 0.73 GAA (0.35) HDAC3CA12CA1IDO1ALOX15
SCHEMBL451924 0.70 HDAC3 (0.54) HDAC3CA12CA1IDO1ALOX15
SCHEMBL7938016 0.70 HDAC3 (0.54) HDAC3CA12CA1IDO1ALOX15
SCHEMBL8219189 0.70 TSHR (0.32) HSD17B10ALDH1A1
SCHEMBL8674456 0.70 ALDH1A1 (0.36) HDAC3CA12CA1IDO1ALOX15
SCHEMBL8675774 0.70 NPC1 (0.38) HDAC3CA12CA1IDO1ALOX15
SCHEMBL10218967 0.69 KMT2A (0.47) HDAC3CA12CA1IDO1ALOX15
SCHEMBL8464352 0.68
SCHEMBL28641832 0.66 HDAC3 (0.58) HDAC3CA12CA1IDO1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0750625-B1 PREPARATION OF MONOCYCLOPENTADIENYL METAL COMPLEXES BY NUCLEOPHILIC SUBSTITUTION OF BIS(CYCLOPENTADIENYL) METAL COMPLEXES DOW CHEMICAL CO (US) 1999-02-03 EP disclosed
US-5659054-A Preparation of monocyclopentadienyl metal complexes by nucleophilic substitution of bis(cyclopentadienyl) metal complexes THE DOW CHEMICAL COMPANY (US) 1997-08-19 US disclosed
EP-0750625-A1 PREPARATION OF MONOCYCLOPENTADIENYL METAL COMPLEXES BY NUCLEOPHILIC SUBSTITUTION OF BIS(CYCLOPENTADIENYL) METAL COMPLEXES THE DOW CHEMICAL COMPANY (US) 1997-01-02 EP disclosed
US-5504224-A Preparation of monocyclopentadienyl metal complexes by nucleophilic substitution of bis(cyclopentadienyl) metal complexes THE DOW CHEMICAL COMPANY (US) 1996-04-02 US disclosed
WO-1995025112-A1 PREPARATION OF MONOCYCLOPENTADIENYL METAL COMPLEXES BY NUCLEOPHILIC SUBSTITUTION OF BIS(CYCLOPENTADIENYL) METAL COMPLEXES THE DOW CHEMICAL COMPANY (US) 1995-09-21 WO disclosed