SCHEMBL8467925

SCHEMBL8467925

Fc1ccc2c(C3CC[N]CC3)nsc2c1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 1/20 0.42
HTR1B P28222 1/20 0.42
GRM4 Q14833 7/20 0.40
CYP1A2 P05177 3/20 0.40
ACHE P22303 2/20 0.33
DRD2 P14416 2/20 0.32
SLC6A4 P31645 1/20 0.32
ALDH1A1 P00352 2/20 0.32
LMNA P02545 1/20 0.32
POLB P06746 1/20 0.32
MAPT P10636 1/20 0.32
RAB9A P51151 3/20 0.32
DRD4 P21917 1/20 0.31
DRD3 P35462 1/20 0.31
GRM2 Q14416 1/20 0.31
SCD O00767 1/20 0.31
NPC1 O15118 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1545776 0.84 CYP1A2 (0.41) HTR1DHTR1BGRM4CYP1A2SLC6A4
Hydrochloric Acid SCHEMBL6221807 0.82 CYP1A2 (0.41) HTR1DHTR1BGRM4CYP1A2SLC6A4
SCHEMBL9429569 0.78 HTR1D (0.38) HTR1DHTR1BGRM4CYP1A2SLC6A4
SCHEMBL3902898 0.78 HTR1D (0.46) HTR1DHTR1BGRM4CYP1A2ACHE
SCHEMBL13898982 0.78 HTR1D (0.44) HTR1DHTR1BGRM4CYP1A2ACHE
SCHEMBL8716257 0.78 HTR1D (0.51) HTR1DHTR1BACHEDRD2SLC6A4
SCHEMBL2204018 0.78 DRD2 (0.46) GRM4CYP1A2ACHEDRD2ALDH1A1
SCHEMBL8678218 0.76 HTR1D (0.37) HTR1DHTR1BGRM4CYP1A2DRD2
SCHEMBL8346568 0.76 HTR1D (0.45) HTR1DHTR1BGRM4CYP1A2ACHE
SCHEMBL6186847 0.76 HTR1D (0.54) HTR1DHTR1BACHEDRD2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5532240-A ANTIPSYCHOTIC AGENTS AND ANTISEROTONIN AGENTS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-07-02 US claimed
US-5874435-A PSYCHOLOGICAL DISORDERS; ANALGESICS HOECHST MARION ROUSSEL, INC. (US) 1999-02-23 US disclosed
US-5854243-A 3-heteroaryl-1-pyrrolidinealkylthiols and derivatives thereof and their therapeutic utility HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1998-12-29 US disclosed
US-5843949-A 1-(1H-indolyloxyalkyl)-4-(heteroaryl)piperazines and related compounds useful as antipsychotics and analgesics HOECHST MARION ROUSSEL, INC. 1998-12-01 US disclosed
US-5840727-A ANTIPSYCHOTICS, ANALGESICS AVENTIS PHARMACEUTICALS INC. 1998-11-24 US disclosed
US-5776963-A ANTIPSYCHOTIC AGENTS HOECHST MARION ROUSSEL, INC. (US) 1998-07-07 US disclosed
US-5691330-A ANTIPSYCHOTIC AGENT YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-11-25 US disclosed
US-5532240-A ANTIPSYCHOTIC AGENTS AND ANTISEROTONIN AGENTS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-07-02 US disclosed