Dipivefrin

Dipivefrin

SCHEMBL8468680

CNCC(O)c1ccc(OC(=O)C(C)(C)C)c(OC(=O)C(C)(C)C)c1.[Li]C(C)CC

nearest known ligand 0.86

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3

The experimentally established mechanism targets of Dipivefrin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 known ✓ P07550 6/20 0.84
ADRA2A known ✓ P08913 4/20 0.42
ADRA2C known ✓ P18825 4/20 0.42
ADRB1 known ✓ P08588 3/20 0.42
ADRB3 known ✓ P13945 3/20 0.42
ADRA2B known ✓ P18089 3/20 0.42
ADRA1A known ✓ P35348 3/20 0.42
ADRA1B known ✓ P35368 2/20 0.42
ADRA1D known ✓ P25100 1/20 0.42
HIF1A Q16665 6/20 0.86
ALDH1A1 P00352 3/20 0.86
CYP3A4 P08684 2/20 0.86
LMNA P02545 2/20 0.86
KDM4E B2RXH2 6/20 0.42
TDP1 Q9NUW8 5/20 0.42
MAPT P10636 3/20 0.42
HSD17B10 Q99714 3/20 0.42
TSHR P16473 3/20 0.42
DRD1 P21728 3/20 0.42
DRD3 P35462 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dipivefrin SCHEMBL24713 0.93 HIF1A (1.00) HIF1AALDH1A1CYP3A4LMNAADRB2
Dipivefrin SCHEMBL29710905 0.93 HIF1A (1.00) HIF1AALDH1A1CYP3A4LMNAADRB2
Dipivefrin SCHEMBL20673238 0.93 HIF1A (1.00) HIF1AALDH1A1CYP3A4LMNAADRB2
Dipivefrin SCHEMBL24714 0.93 HIF1A (1.00) HIF1AALDH1A1CYP3A4LMNAADRB2
Dipivefrin SCHEMBL5275338 0.91 ADRB2 (1.00) HIF1AALDH1A1CYP3A4LMNAADRB2
Dipivefrin SCHEMBL41350 0.91 ADRB2 (1.00) HIF1AALDH1A1CYP3A4LMNAADRB2
Dipivefrin SCHEMBL41351 0.91 ADRB2 (1.00) HIF1AALDH1A1CYP3A4LMNAADRB2
Dipivefrin SCHEMBL8071336 0.91 ADRB2 (1.00) HIF1AALDH1A1CYP3A4LMNAADRB2
Dipivefrin SCHEMBL18687014 0.91 ADRB2 (1.00) HIF1AALDH1A1CYP3A4LMNAADRB2
Dipivefrin SCHEMBL3053588 0.90 HIF1A (0.95) HIF1AALDH1A1CYP3A4LMNAADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5955546-A COATING POLYPROPYLENE OR ETHYLENE/ALPHA-OLEFIN COPOLYMER HAVING A PRIMARY POLYOLEFIN SEGMENT LENGTH WITHIN A RANGE OF ABSOLUTE VALUE OF FROM ABOUT 4.2 TO ABOUT 8.8, WITH AT LEAST ONE MODIFYING POLYOLEFIN COMPRISING A COPOLYMER OF ETHYLENE REGENTS OF THE UNIVERSITY OF MINNESOTA 1999-09-21 US disclosed
US-5710219-A Miscible polyolefin blends REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 1998-01-20 US disclosed
US-5654364-A Miscible blend of polyolefin and polyolefin block copolymer REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 1997-08-05 US disclosed
US-5571864-A POLYPROPYLENE BLENDED WITH ETHYLENE OR OLEFIN POLYMER OR BLOCK POLYMER REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 1996-11-05 US disclosed
EP-0620251-A2 Miscible polyolefin blends REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 1994-10-19 EP disclosed