SCHEMBL8469459

SCHEMBL8469459

CN(C)c1ncc2cc([N+](=O)[O-])ccc2n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
CYP1A2 P05177 2/20 0.45
HTT P42858 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
CDK1 P06493 1/20 0.43
CCNB1 P14635 1/20 0.43
CCNE1 P24864 1/20 0.43
CDK2 P24941 1/20 0.43
CYP3A4 P08684 1/20 0.43
NAMPT P43490 1/20 0.43
XDH P47989 1/20 0.43
MAPT P10636 3/20 0.42
POLB P06746 1/20 0.42
MAOB P27338 1/20 0.42
NOS1 P29475 1/20 0.42
TXNRD1 Q16881 1/20 0.41
TXNRD3 Q86VQ6 1/20 0.41
TXNRD2 Q9NNW7 1/20 0.41
KMT2A Q03164 2/20 0.41
TDP1 Q9NUW8 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ammonia Solution, Strong SCHEMBL8471114 0.98 ALDH1A1 (0.45) ALDH1A1CYP1A2HTTSMN1; SMN2CDK1
SCHEMBL4535746 0.80 SMN1; SMN2 (0.50) ALDH1A1CYP1A2HTTSMN1; SMN2CDK1
SCHEMBL31155580 0.80 SMN1; SMN2 (0.50) ALDH1A1CYP1A2HTTSMN1; SMN2CDK1
SCHEMBL27456953 0.78 CYP1A2 (0.42) ALDH1A1CYP1A2HTTSMN1; SMN2CDK1
SCHEMBL27920418 0.76 ALDH1A1 (0.46) ALDH1A1CYP1A2HTTSMN1; SMN2CYP3A4
SCHEMBL1438547 0.76 MAPT (0.51) ALDH1A1CYP1A2CYP3A4NAMPTXDH
SCHEMBL27350722 0.76 KMT2A (0.51) ALDH1A1CYP1A2HTTSMN1; SMN2CYP3A4
SCHEMBL11150396 0.76 TXNRD1 (0.49) ALDH1A1CYP1A2SMN1; SMN2CYP3A4NAMPT
SCHEMBL27981594 0.76 ALDH1A1 (0.46) ALDH1A1CYP1A2HTTSMN1; SMN2CYP3A4
SCHEMBL24207471 0.76 KDM4E (0.45) ALDH1A1CYP1A2HTTSMN1; SMN2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0892789-A1 IRREVERSIBLE INHIBITORS OF TYROSINE KINASES WARNER-LAMBERT COMPANY (US) 1999-01-27 EP disclosed
WO-1997038983-A1 IRREVERSIBLE INHIBITORS OF TYROSINE KINASES WARNER-LAMBERT COMPANY (US) 1997-10-23 WO disclosed