SCHEMBL8470385

SCHEMBL8470385

O=C1c2ccccc2OCC1SC(=O)C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 15/20 0.47
MAOB P27338 2/20 0.43
SIGMAR1 Q99720 1/20 0.37
PKM P14618 1/20 0.37
TSHR P16473 1/20 0.37
HDAC1 Q13547 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8473045 0.85 CYP19A1 (0.41) CYP19A1MAOB
SCHEMBL8472084 0.84 CYP19A1 (0.40) CYP19A1MAOB
SCHEMBL8470417 0.84 CYP19A1 (0.50) CYP19A1MAOB
SCHEMBL8472750 0.81 CYP19A1 (0.53) CYP19A1
SCHEMBL7294129 0.77 CYP19A1 (0.56) CYP19A1MAOBSIGMAR1PKMTSHR
SCHEMBL8470409 0.77 CYP19A1 (0.49) CYP19A1MAOBSIGMAR1PKMTSHR
SCHEMBL8470905 0.76 CYP19A1 (0.34) CYP19A1
SCHEMBL9835237 0.73 CYP19A1 (0.56) CYP19A1MAOBSIGMAR1PKMTSHR
SCHEMBL9094361 0.73 CYP19A1 (0.56) CYP19A1MAOBSIGMAR1PKMTSHR
SCHEMBL7153929 0.73 CYP19A1 (0.56) CYP19A1MAOBSIGMAR1PKMTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5886016-A ANTIINFLAMMATORY AGENT WITH MINIMAL SIDE EFFECTS FOR TREATING ARTHRITIS G.D. SEARLE & CO. (US) 1999-03-23 US disclosed
US-5670532-A Pyrazolyl derivatives for the treatment of inflammation G. D. SEARLE & CO. (US) 1997-09-23 US disclosed
US-5565482-A ANTIINFLAMMATORY AGENTS, ANTIARTHRITIC AGENTS G.D. SEARLE & CO. (US) 1996-10-15 US disclosed
US-5547975-A ANTIARTHRIC AGENTS, ANALGESICS AND ANTIPYRETICS; INHIBITORS OF CYCLOOXYGENASE II; SIDE EFFECT REDUCTION G.D. SEARLE & CO. 1996-08-20 US disclosed
WO-1996009304-A1 BENZOPYRANOPYRAZOLYL DERIVATIVES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-03-28 WO disclosed