SCHEMBL8470409

SCHEMBL8470409

O=C1c2ccccc2OCC1C(=O)C(F)(F)F

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 15/20 0.49
MAOB P27338 2/20 0.46
HDAC1 Q13547 1/20 0.40
PKM P14618 1/20 0.39
TSHR P16473 1/20 0.39
SIGMAR1 Q99720 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7840882 0.81 CYP19A1 (0.46) CYP19A1MAOBHDAC1PKMTSHR
SCHEMBL8470357 0.81 CYP19A1 (0.52) CYP19A1MAOB
SCHEMBL3520052 0.81 CYP19A1 (0.58) CYP19A1MAOBPKMTSHRSIGMAR1
SCHEMBL11635929 0.80 CYP19A1 (0.53) CYP19A1MAOBPKMTSHRSIGMAR1
SCHEMBL11424192 0.78 CYP19A1 (0.48) CYP19A1MAOBPKMTSHRSIGMAR1
Fluoride SCHEMBL11424190 0.77 CYP19A1 (0.50) CYP19A1MAOBPKMTSHRSIGMAR1
SCHEMBL8470385 0.77 CYP19A1 (0.47) CYP19A1MAOBHDAC1PKMTSHR
SCHEMBL31336705 0.74 CYP19A1 (0.54) CYP19A1MAOBPKMTSHRSIGMAR1
SCHEMBL9832882 0.74 MAOB (0.47) CYP19A1MAOBHDAC1SIGMAR1
SCHEMBL28699476 0.73 KDM4E (0.51) CYP19A1HDAC1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5886016-A ANTIINFLAMMATORY AGENT WITH MINIMAL SIDE EFFECTS FOR TREATING ARTHRITIS G.D. SEARLE & CO. (US) 1999-03-23 US disclosed
US-5670532-A Pyrazolyl derivatives for the treatment of inflammation G. D. SEARLE & CO. (US) 1997-09-23 US disclosed
US-5565482-A ANTIINFLAMMATORY AGENTS, ANTIARTHRITIC AGENTS G.D. SEARLE & CO. (US) 1996-10-15 US disclosed
US-5547975-A ANTIARTHRIC AGENTS, ANALGESICS AND ANTIPYRETICS; INHIBITORS OF CYCLOOXYGENASE II; SIDE EFFECT REDUCTION G.D. SEARLE & CO. 1996-08-20 US disclosed
WO-1996009304-A1 BENZOPYRANOPYRAZOLYL DERIVATIVES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-03-28 WO disclosed