SCHEMBL8470436

SCHEMBL8470436

CC(COC=O)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRIA4 P48058 1/20 0.46
PTGS2 P35354 1/20 0.44
CHRNB2 P17787 1/20 0.39
CHRNA4 P43681 1/20 0.39
CYP1A2 P05177 1/20 0.38
GAA P10253 1/20 0.38
CYP2C9 P11712 1/20 0.38
PKM P14618 1/20 0.38
CYP2C19 P33261 1/20 0.38
PDCD1 Q15116 1/20 0.38
CD274 Q9NZQ7 1/20 0.38
TAAR1 Q96RJ0 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL424240 0.89 TAAR1 (0.47) TAAR1
SCHEMBL23315604 0.79 TYR (0.31)
SCHEMBL2312796 0.77 GRIA4 (0.50) GRIA4PTGS2CHRNB2CHRNA4TAAR1
SCHEMBL8470432 0.76 GRIA4 (0.46) GRIA4PTGS2CHRNB2CHRNA4CYP1A2
SCHEMBL4309371 0.73 APP (0.39) CYP1A2
SCHEMBL11609177 0.73 GRIA4 (0.48) GRIA4PTGS2
SCHEMBL528539 0.73 CYP1A2 (0.56) GRIA4PTGS2CYP1A2GAACYP2C9
SCHEMBL20563823 0.73 CYP1A2 (0.56) GRIA4PTGS2CYP1A2GAACYP2C9
SCHEMBL1966503 0.73 KCNJ1 (0.44) PTGS2CYP1A2GAA
SCHEMBL9572888 0.71 RIPK1 (0.47) TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4520193-A Cephalosporin derivatives RHONE-POULENC INDUSTRIES (FR) 1985-05-28 US claimed
US-5952497-A USEFUL IN PEPTIDE, POLYPEPTIDE AND PROTEIN SYNTHESIS UNIVERSITY OF GEORGIA RESEARCH FOUNDATION (US) 1999-09-14 US disclosed